Suzuki-Miyaura cross-coupling reactions of potassium Boc-protected aminomethyltrifluoroborate with aryl and hetaryl mesylates

Org Lett. 2012 Jun 15;14(12):3138-41. doi: 10.1021/ol301221p. Epub 2012 May 31.

Abstract

Palladium-catalyzed Suzuki-Miyaura cross-coupling reactions were studied with potassium Boc-protected aminomethyltrifluoroborate through C-O activation of various mesylate derivatives to afford the corresponding products in moderate to good yields.

Publication types

  • Research Support, N.I.H., Extramural

MeSH terms

  • Amination
  • Boric Acids / chemistry*
  • Fluorine Compounds / chemistry*
  • Mesylates / chemistry*
  • Methylation
  • Molecular Structure
  • Oxidation-Reduction
  • Potassium / chemistry*

Substances

  • Boric Acids
  • Fluorine Compounds
  • Mesylates
  • boric acid
  • Potassium