M-opsin protein degradation is inhibited by MG-132 in Rpe65⁻/⁻ retinal explant culture

Mol Vis. 2012:18:1516-25. Epub 2012 Jun 13.

Abstract

Purpose: The 65 kDa retinal pigment epithelium-specific protein, RPE65, is an essential enzyme for 11-cis-retinal synthesis in the eye. Mutations of the RPE65 gene in humans result in severe vision loss, and Rpe65(-/-) mice show early cone photoreceptor degeneration. We used an explant culture system to evaluate whether posttranslational downregulation of M-opsin protein in Rpe65(-/-) mice is caused by proteolytic degradation.

Methods: The eyes of three-week-old Rpe65(-/-) mice were incubated in culture medium. Western blot analysis was used to evaluate the level of M-opsin protein, and immunofluorescence was used for protein localization. The transcriptional level of M-opsin was evaluated with real-time reverse-transcriptase-PCR.

Results: Degradation of the M-opsin protein in Rpe65(-/-) mouse retina was inhibited by the proteasome inhibitor MG-132 but not by the lysosomal inhibitor pepstatin A and E64d. 9-cis-retinal, used as an analog of 11-cis-retinal, increased M-opsin protein but did not increase M-opsin mRNA. Moreover, 9-cis-retinal did not change the transcriptional levels of photoreceptor specific genes.

Conclusions: Our data suggest that M-opsin protein was degraded through a proteasome pathway and that M-opsin degradation was suppressed with 9-cis-retinal treatment in Rpe65(-/-) mice to some extent.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Cone Opsins / genetics
  • Cone Opsins / metabolism*
  • Cysteine Proteinase Inhibitors / pharmacology
  • Diterpenes
  • Eye / drug effects*
  • Eye / metabolism
  • Leucine / analogs & derivatives
  • Leucine / pharmacology
  • Leupeptins / pharmacology*
  • Lysosomes / metabolism
  • Mice
  • Mice, Knockout
  • Organ Culture Techniques
  • Pepstatins / pharmacology
  • Proteasome Endopeptidase Complex / metabolism
  • Proteasome Inhibitors*
  • Proteolysis / drug effects
  • Real-Time Polymerase Chain Reaction
  • Retinaldehyde / pharmacology
  • Transcription, Genetic / drug effects
  • cis-trans-Isomerases / deficiency
  • cis-trans-Isomerases / genetics*

Substances

  • Cone Opsins
  • Cysteine Proteinase Inhibitors
  • Diterpenes
  • Leupeptins
  • Pepstatins
  • Proteasome Inhibitors
  • 9-cis-retinal
  • retinoid isomerohydrolase
  • Proteasome Endopeptidase Complex
  • cis-trans-Isomerases
  • Leucine
  • aloxistatin
  • benzyloxycarbonylleucyl-leucyl-leucine aldehyde
  • Retinaldehyde
  • pepstatin