Voltage-sensing phosphatase reveals temporal regulation of TRPC3/C6/C7 channels by membrane phosphoinositides

Channels (Austin). 2012 May-Jun;6(3):206-9. doi: 10.4161/chan.20883. Epub 2012 May 1.

Abstract

TRPC3/C6/C7 channels, a subgroup of classical/canonical TRP channels, are activated by diacylglycerol produced via activation of phospholipase C (PLC)-coupled receptors. Recognition of the physiological importance of these channels has been steadily growing, but the mechanism by which they are regulated remains largely unknown. We recently used a membrane-resident danio rerio voltage-sensing phosphatase (DrVSP) to study TRPC3/C6/C7 regulation and found that the channel activity was controlled by PtdIns(4,5)P(2)-DAG signaling in a self-limiting manner (Imai Y et al., the Journal of Physiology, 2012). In this addendum, we present the advantages of using DrVSP as a molecular tool to study PtdIns(4,5)P(2) regulation. DrVSP should be readily applicable for studying phosphoinositide metabolism-linked channel regulation as well as lipid dynamics. Furthermore, in comparison to other modes of self-limiting ion channel regulation, the regulation of TRPC3/C6/C7 channels seems highly susceptible to activation signal strength, which could potentially affect both open duration and the time to peak activation and inactivation. Dysfunction of such self-limiting regulation may contribute to the pathology of the cardiovascular system, gastrointestinal tract and brain, as these channels are broadly distributed and affected by numerous neurohormonal agonists.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Cell Line, Transformed
  • Ciona intestinalis
  • Diglycerides / metabolism
  • Humans
  • Ion Channel Gating
  • Mice
  • Phosphatidylinositol 4,5-Diphosphate / metabolism
  • Phosphoinositide Phospholipase C / metabolism
  • Phosphoric Monoester Hydrolases / metabolism*
  • Species Specificity
  • TRPC Cation Channels / metabolism*
  • TRPC6 Cation Channel
  • Zebrafish Proteins / metabolism*

Substances

  • Diglycerides
  • Phosphatidylinositol 4,5-Diphosphate
  • TRPC Cation Channels
  • TRPC3 cation channel
  • TRPC6 Cation Channel
  • TRPC6 protein, human
  • Trpc7 protein, mouse
  • Zebrafish Proteins
  • tpte protein, zebrafish
  • voltage-sensor-containing phosphatase, Ciona intestinalis
  • Phosphoric Monoester Hydrolases
  • Phosphoinositide Phospholipase C