The effects of 17β-estradiol plus drospirenone on anthropometric and biochemical measures of adiposity in menopausal women

Arch Gynecol Obstet. 2012 Nov;286(5):1233-9. doi: 10.1007/s00404-012-2437-9. Epub 2012 Jul 13.

Abstract

Purpose: To assess whether there are changes on anthropometric and biochemical measures of adiposity in pre- and postmenopausal women and in the latter before and after 6 months treatment with 17β-estradiol plus drospirenone.

Methods: Twenty postmenopausal and 20 premenopausal women were enrolled in a prospective comparative study. Postmenopausal women received 1 mg 17β-estradiol plus 2 mg drospirenone daily for 6 months. Measurements of body mass index (BMI), waist/hip ratio and plasmatic levels of insulin, glucose, high-density lipoprotein (HDL), low-density lipoprotein (LDL), triglyceride, leptin, adiponectin, orexin-A, glucagon-like peptide-1 (GLP-1) and ghrelin were performed in premenopausal (group 1) and postmenopausal women and in the latter before (group 2a) and after (group 2b) 6 months treatment with 17β-estradiol plus drospirenone.

Results: No significant changes in BMIs, insulin and glucose were observed between group 1 and 2a; and group 2a and 2b. GLP-1 levels were significantly increased in group 1 compared to group 2a (p = 0.035). Leptin levels were significantly increased (p = 0.001) and GLP-1 levels were significantly decreased (p = 0.021) in group 2b compared to group 2a. HDL was significantly decreased while LDL and triglyceride levels were significantly increased in group 2a compared to group 1. (p = 0.030, p = 0.001, p = 0.020; respectively) LDL was significantly decreased (p = 0.010) in group 2b compared to group 2a. GLP-1 had a positive correlation with orexin-A (p < 0.001, r = 0.520) and negative correlation with leptin (p = 0.008, r = -0.345).

Conclusion: Leptin was significantly higher and GLP-1 was significantly lower in women receiving 17β-estradiol plus drospirenone treatment. GLP-1 levels were significantly lower after the menopause compared to premenopausal levels. Orexin-A and GLP-1 were positively correlated.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Adiponectin / blood
  • Adiposity / drug effects*
  • Adult
  • Androstenes / pharmacology*
  • Blood Glucose / metabolism
  • Body Mass Index
  • Drug Therapy, Combination
  • Estradiol / pharmacology*
  • Estrogen Replacement Therapy
  • Estrogens / pharmacology
  • Female
  • Ghrelin / blood
  • Glucagon-Like Peptide 1 / blood
  • Humans
  • Insulin / blood
  • Intracellular Signaling Peptides and Proteins / blood
  • Leptin / blood
  • Lipoproteins, HDL / blood
  • Lipoproteins, LDL / blood
  • Middle Aged
  • Mineralocorticoid Receptor Antagonists / pharmacology
  • Neuropeptides / blood
  • Orexins
  • Postmenopause / blood
  • Postmenopause / physiology*
  • Premenopause / blood
  • Premenopause / physiology*
  • Triglycerides / blood
  • Waist-Hip Ratio

Substances

  • Adiponectin
  • Androstenes
  • Blood Glucose
  • Estrogens
  • Ghrelin
  • HCRT protein, human
  • Insulin
  • Intracellular Signaling Peptides and Proteins
  • Leptin
  • Lipoproteins, HDL
  • Lipoproteins, LDL
  • Mineralocorticoid Receptor Antagonists
  • Neuropeptides
  • Orexins
  • Triglycerides
  • Estradiol
  • Glucagon-Like Peptide 1
  • drospirenone