Effect of β-blocker cessation on chronotropic incompetence and exercise tolerance in patients with advanced heart failure

Circ Heart Fail. 2012 Sep 1;5(5):560-5. doi: 10.1161/CIRCHEARTFAILURE.112.967695. Epub 2012 Aug 1.

Abstract

Background: Chronotropic incompetence is defined as the inability to reach 80% of heart rate (HR) reserve or 80% of the maximally predicted HR during exercise. The presence of chronotropic incompetence is associated with reduced peak oxygen consumption, and rate-responsive pacing therapy is under investigation to improve exercise capacity in heart failure (HF). However, uncertainty exists about whether chronotropic incompetence and reduced exercise tolerance in HF are attributable to β-blockade.

Methods and results: Subjects with HF and receiving long-term β-blocker therapy underwent cardiopulmonary exercise tolerance testing under 2 conditions in random sequence: (1) after a 27-hour washout period (Off-BB) and (2) 3 hours after β-blocker ingestion (On-BB). Norepinephrine levels were drawn at rest and at peak exercise. β1-response to norepinephrine was assessed using the chronotropic responsiveness index: ΔHR/Δlog norepinephrine. Nineteen patients with systolic HF (left ventricular ejection fraction, 22.8±7.7%) were enrolled. Mean age was 49.4±12.3 years. Average carvedilol equivalent dose was 29.1±17.0 mg daily. Peak HR off/on β-blockers was 62.7±18.7% and 51.4±18.2% HR reserve (P<0.01) and 79.1±11.0% and 70.3±12.3% maximally predicted HR (P<0.01). For the Off-BB and On-BB conditions, the respiratory exchange ratios were 1.05±0.06 and 1.05±0.10 (P=0.77), respectively, confirming maximal and near identical effort in both conditions. The peak oxygen consumption was 16.6±3.34 and 15.9±3.31 mL/kg/min (P=0.03), and the chronotropic responsiveness index was 19.3±7.2 and 16.2±7.1 (P=0.18).

Conclusions: Acute β-blocker cessation does not normalize the chronotropic response to exercise in patients with advanced HF and chronotropic incompetence.

Publication types

  • Randomized Controlled Trial
  • Research Support, N.I.H., Extramural

MeSH terms

  • Adrenergic beta-Antagonists / administration & dosage*
  • Adult
  • Analysis of Variance
  • Biomarkers / blood
  • Bisoprolol / administration & dosage
  • Carbazoles / administration & dosage
  • Carvedilol
  • Drug Administration Schedule
  • Exercise Test
  • Exercise Tolerance / drug effects*
  • Female
  • Heart Failure / blood
  • Heart Failure / diagnosis
  • Heart Failure / drug therapy*
  • Heart Failure / physiopathology
  • Heart Rate / drug effects*
  • Humans
  • Male
  • Metoprolol / administration & dosage
  • Middle Aged
  • New York City
  • Norepinephrine / blood
  • Oxygen Consumption / drug effects
  • Propanolamines / administration & dosage
  • Prospective Studies
  • Respiration / drug effects
  • Time Factors

Substances

  • Adrenergic beta-Antagonists
  • Biomarkers
  • Carbazoles
  • Propanolamines
  • Carvedilol
  • Metoprolol
  • Norepinephrine
  • Bisoprolol