ADP ribosylation adapts an ER chaperone response to short-term fluctuations in unfolded protein load

J Cell Biol. 2012 Aug 6;198(3):371-85. doi: 10.1083/jcb.201202005.

Abstract

Gene expression programs that regulate the abundance of the chaperone BiP adapt the endoplasmic reticulum (ER) to unfolded protein load. However, such programs are slow compared with physiological fluctuations in secreted protein synthesis. While searching for mechanisms that fill this temporal gap in coping with ER stress, we found elevated levels of adenosine diphosphate (ADP)-ribosylated BiP in the inactive pancreas of fasted mice and a rapid decline in this modification in the active fed state. ADP ribosylation mapped to Arg470 and Arg492 in the substrate-binding domain of hamster BiP. Mutations that mimic the negative charge of ADP-ribose destabilized substrate binding and interfered with interdomain allosteric coupling, marking ADP ribosylation as a rapid posttranslational mechanism for reversible inactivation of BiP. A kinetic model showed that buffering fluctuations in unfolded protein load with a recruitable pool of inactive chaperone is an efficient strategy to minimize both aggregation and costly degradation of unfolded proteins.

Publication types

  • Research Support, N.I.H., Extramural
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Adenosine Diphosphate / chemistry*
  • Allosteric Site
  • Animals
  • Anisotropy
  • Catalytic Domain
  • Cell Line
  • Cricetinae
  • Endoplasmic Reticulum / metabolism*
  • Endoplasmic Reticulum Chaperone BiP
  • Heat-Shock Proteins / metabolism
  • Heat-Shock Proteins / physiology*
  • Homeostasis
  • Humans
  • Kinetics
  • Mice
  • Molecular Chaperones
  • Mutation
  • Protein Denaturation
  • Protein Folding
  • Proteins / chemistry*
  • Ribose / chemistry

Substances

  • Endoplasmic Reticulum Chaperone BiP
  • Heat-Shock Proteins
  • Molecular Chaperones
  • Proteins
  • Adenosine Diphosphate
  • Ribose