In vivo effect of glucose-dependent insulinotropic peptide (GIP) on the gene expression of calcitonin peptides in human subcutaneous adipose tissue

Regul Pept. 2012 Nov 10;179(1-3):29-32. doi: 10.1016/j.regpep.2012.08.004. Epub 2012 Sep 5.

Abstract

Background: Increased plasma levels of calcitonin gene-related peptide-I (CGRP-I) and procalcitonin (Pro-CT) (both also named calcitonin peptides (CT peptides)) are associated with obesity and systemic inflammation. Glucose-dependent insulinotropic polypeptide (GIP), a nutrient-dependent incretin hormone, was recently found to induce CGRP-I and CT expression in human adipocytes in vitro. However, a physiological relevance of a possible interaction between GIP and CT peptides has not yet been studied.

Methods: In this study, we analyzed the effect of GIP on the expression of CGRP-I and CT mRNA in human subcutaneous adipose tissue within a randomized, controlled trial. Seventeen male obese subjects were infused with GIP [2.0 pmol kg(-1) min(-1) for 240 min] or placebo, either in the fasting state, during euglycemic-hyperinsulinemic (EC) or hyperglycemic-hyperinsulinemic clamps (HC).

Results: The CGRP-I gene expression was detected in all investigated adipose tissue samples, whereas very low CT expression was found in only 8 out of 116 analyzed samples. No significant influence of either GIP or glucose and insulin infusions on the CGRP-I and CT expression was observed in any of the individual experiments (GIP infusion, EC and HC) or in the combined analysis of all experiments with and without GIP. Furthermore, CGRP-I expression was not correlated with plasma GIP level before or after 240 min of infusions or clamps.

Conclusion: In contrast to in vitro data, an acute application of GIP has no effect on mRNA expression of CT peptides in subcutaneous adipose tissue of obese humans.

Publication types

  • Randomized Controlled Trial
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Adult
  • Blood Glucose
  • Calcitonin / blood*
  • Calcitonin / genetics
  • Calcitonin Gene-Related Peptide
  • Gastric Inhibitory Polypeptide / blood
  • Gastric Inhibitory Polypeptide / pharmacology*
  • Gene Expression Regulation*
  • Glucose Clamp Technique / methods
  • Humans
  • Hyperinsulinism / metabolism
  • Insulin / blood
  • Male
  • Middle Aged
  • Obesity / genetics
  • Obesity / metabolism*
  • Protein Precursors / blood*
  • Protein Precursors / genetics
  • RNA, Messenger / genetics
  • RNA, Messenger / metabolism
  • Subcutaneous Fat / drug effects
  • Subcutaneous Fat / metabolism*
  • Waist-Hip Ratio

Substances

  • Blood Glucose
  • CALCA protein, human
  • Insulin
  • Protein Precursors
  • RNA, Messenger
  • Gastric Inhibitory Polypeptide
  • Calcitonin
  • Calcitonin Gene-Related Peptide