Microneedle mediated intradermal delivery of adjuvanted recombinant HIV-1 CN54gp140 effectively primes mucosal boost inoculations

J Control Release. 2012 Sep 28;162(3):529-37. doi: 10.1016/j.jconrel.2012.07.039. Epub 2012 Aug 7.

Abstract

Dissolving polymeric microneedle arrays formulated to contain recombinant CN54 HIVgp140 and the TLR4 agonist adjuvant MPLA were assessed for their ability to elicit antigen-specific immunity. Using this novel microneedle system we successfully primed antigen-specific responses that were further boosted by an intranasal mucosal inoculation to elicit significant antigen-specific immunity. This prime-boost modality generated similar serum and mucosal gp140-specific IgG levels to the adjuvanted and systemic subcutaneous inoculations. While the microneedle primed groups demonstrated a balanced Th1/Th2 profile, strong Th2 polarization was observed in the subcutaneous inoculation group, likely due to the high level of IL-5 secretion from cells in this group. Significantly, the animals that received a microneedle prime and intranasal boost regimen elicited a high level IgA response in both the serum and mucosa, which was greatly enhanced over the subcutaneous group. The splenocytes from this inoculation group secreted moderate levels of IL-5 and IL-10 as well as high amounts of IL-2, cytokines known to act in synergy to induce IgA. This work opens up the possibility for microneedle-based HIV vaccination strategies that, once fully developed, will greatly reduce risk for vaccinators and patients, with those in the developing world set to benefit most.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • AIDS Vaccines
  • Adjuvants, Immunologic / administration & dosage*
  • Administration, Cutaneous
  • Animals
  • Cytokines / immunology
  • Female
  • HIV-1
  • Immunoglobulin A / blood
  • Immunoglobulin A / immunology
  • Immunoglobulin G / blood
  • Immunoglobulin G / immunology
  • Lipid A / administration & dosage
  • Lipid A / analogs & derivatives*
  • Mice
  • Mice, Inbred BALB C
  • Microinjections*
  • Needles
  • Recombinant Proteins / administration & dosage
  • Spleen / cytology
  • Spleen / immunology
  • Toll-Like Receptor 4 / agonists
  • Vagina / immunology
  • env Gene Products, Human Immunodeficiency Virus / administration & dosage*
  • env Gene Products, Human Immunodeficiency Virus / immunology

Substances

  • AIDS Vaccines
  • Adjuvants, Immunologic
  • Cytokines
  • Immunoglobulin A
  • Immunoglobulin G
  • Lipid A
  • Recombinant Proteins
  • Tlr4 protein, mouse
  • Toll-Like Receptor 4
  • env Gene Products, Human Immunodeficiency Virus
  • gp140 envelope protein, Human immunodeficiency virus 1
  • monophosphoryl lipid A