Antimicrobial photodynamic therapy with RLP068 kills methicillin-resistant Staphylococcus aureus and improves wound healing in a mouse model of infected skin abrasion PDT with RLP068/Cl in infected mouse skin abrasion

J Biophotonics. 2013 Sep;6(9):733-42. doi: 10.1002/jbio.201200121. Epub 2012 Sep 14.

Abstract

Photodynamic therapy (PDT) is an alternative treatment for infections that can kill drug resistant bacteria without damaging host-tissue. In this study we used bioluminescent methicillin-resistant Staphylococcus aureus, in a mouse skin abrasion model, to investigate the effect of PDT on bacterial inactivation and wound healing. RLP068/Cl, a tetracationic Zn(II)phthalocyanine derivative and toluidine blue (TBO) were used. The light-dose response of PDT to kill bacteria in vivo and the possible recurrence in the days post-treatment were monitored by real-time bioluminescence imaging, and wound healing by digital photography. The results showed PDT with RLP068/Cl (but not TBO) was able to kill bacteria, to inhibit bacterial re-growth after the treatment and to significantly accelerate the wound healing process (© 2013 WILEY-VCH Verlag GmbH & Co. KGaA, Weinheim).

Keywords: Antimicrobial photodynamic therapy; cationic zinc phthalocyanine bioluminescence imaging; methicillin resistant Staphylococcus aureus; skin abrasion; skin and soft tissue infection; wound healing.

Publication types

  • Research Support, N.I.H., Extramural
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Anti-Infective Agents / pharmacology*
  • Anti-Infective Agents / therapeutic use
  • Disease Models, Animal
  • Female
  • Indoles / pharmacology*
  • Indoles / therapeutic use
  • Luminescent Measurements
  • Methicillin-Resistant Staphylococcus aureus / drug effects*
  • Methicillin-Resistant Staphylococcus aureus / physiology
  • Mice
  • Mice, Inbred BALB C
  • Organometallic Compounds / pharmacology*
  • Organometallic Compounds / therapeutic use
  • Photochemotherapy*
  • Photosensitizing Agents / pharmacology*
  • Photosensitizing Agents / therapeutic use
  • Staphylococcal Skin Infections / drug therapy*
  • Tolonium Chloride / pharmacology
  • Tolonium Chloride / therapeutic use
  • Wound Healing / drug effects*

Substances

  • Anti-Infective Agents
  • Indoles
  • Organometallic Compounds
  • Photosensitizing Agents
  • RLP068
  • Tolonium Chloride