RNA-protein interaction. An analysis with RNA oligonucleotides of the recognition by alpha-sarcin of a ribosomal domain critical for function

J Biol Chem. 1990 Feb 5;265(4):2216-22.

Abstract

alpha-Sarcin is a cytotoxic protein that inactivates ribosomes by hydrolyzing a single phosphodiester bond on the 3' side of G-4325 in eukaryotic 28 S rRNA. We have examined the requirements for the recognition by alpha-sarcin of this domain using a synthetic oligoribonucleotide (35-mer) that reproduces the sequence and, we presume, the secondary structure (a stem, a bulged nucleotide, and a loop) at the site of modification. The wild type structure and a large number of variants were transcribed in vitro from synthetic DNA templates with phage T7 RNA polymerase. Recognition of the substrate is strongly favored by a G at the position that corresponds to 4325. There is an absolute requirement for a helical stem; however, it can be reduced from the 7 base pairs in the natural structure to 3 without loss of specificity. The nature of the base pairs in the stem modifies but does not abolish recognition; whereas, the bulged nucleotide does not contribute to identification. Cleavage is materially affected by altering the nucleotides in the universal sequence surrounding G-4325 and changing the position in the loop of the tetranucleotide GAG(sarcin)A leads to loss of recognition by the toxin. We propose that the alpha-sarcin domain RNA participates in elongation factor catalyzed binding of aminoacyl-tRNA and of translocation; that translocation is driven by transitions in the structure of the alpha-sarcin domain RNA initiated by the binding of the factors, or the hydrolysis of GTP, or both; and that to toxin inactivates the ribosomes by preventing this transition.

Publication types

  • Research Support, Non-U.S. Gov't
  • Research Support, U.S. Gov't, P.H.S.

MeSH terms

  • Adenosine
  • Aspergillus / metabolism
  • Base Composition
  • Base Sequence
  • Endoribonucleases*
  • Fungal Proteins / metabolism*
  • Molecular Sequence Data
  • Nucleic Acid Conformation
  • Oligoribonucleotides / metabolism*
  • Protein Binding
  • Protein Synthesis Inhibitors / metabolism
  • RNA, Ribosomal, 28S / metabolism
  • Structure-Activity Relationship
  • Substrate Specificity

Substances

  • Fungal Proteins
  • Oligoribonucleotides
  • Protein Synthesis Inhibitors
  • RNA, Ribosomal, 28S
  • alpha-sarcin
  • Endoribonucleases
  • Adenosine