Serum- and glucocorticoid-inducible kinase SGK1 regulates reorganization of actin cytoskeleton in mast cells upon degranulation

Am J Physiol Cell Physiol. 2013 Jan 1;304(1):C49-55. doi: 10.1152/ajpcell.00179.2012. Epub 2012 Sep 26.

Abstract

Aggregation of the high-affinity IgE receptor (FcεRI) on mast cells (MCs) causes MC degranulation, a process that involves cortical F-actin disassembly. Actin depolymerization may be triggered by increase of cytosolic Ca(2+). Entry of Ca(2+) through the Ca(2+) release-activated Ca(2+) (CRAC) channels is under powerful regulation by the serum- and glucocorticoid-inducible kinase SGK1. Moreover, FcεRI-dependent degranulation is decreased in SGK1-deficient (sgk1(-/-)) MCs. The present study addressed whether SGK1 is required for actin cytoskeleton rearrangement in MCs and whether modulation of actin architecture could underlie decreased degranulation of sgk1(-/-) MCs. Confirming previous results, release of β-hexosaminidase reflecting FcεRI-dependent degranulation was impaired in sgk1(-/-) MCs compared with sgk1(+/+) MCs. When CRAC channels were inhibited by 2-aminoethoxydiphenyl borate (2-APB; 50 μM), MC degranulation was strongly decreased in both sgk1(+/+) and sgk1(-/-) MCs and the difference between genotypes was abolished. Moreover, degranulation was impaired by actin-stabilizing (phallacidin) and enhanced by actin-disrupting (cytochalasin B) agents to a similar extent in sgk1(+/+) MCs and sgk1(-/-) MCs, implying a regulatory role of actin reorganization in this event. In line with this, measurements of monomeric (G) and filamentous (F) actin content by FACS analysis and Western blotting of detergent-soluble and -insoluble cell fractions indicated an increase of the G/F-actin ratio in sgk1(+/+) MCs but not in sgk1(-/-) MCs upon FcεRI ligation, an observation reflecting actin depolymerization. In sgk1(+/+) MCs, FcεRI-induced actin depolymerization was abolished by 2-APB. The observed actin reorganization was confirmed by confocal laser microscopic analysis. Our observations uncover SGK1-dependent Ca(2+) entry in mast cells as a novel mechanism regulating actin cytoskeleton.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Actin Cytoskeleton / drug effects
  • Actin Cytoskeleton / enzymology*
  • Actins / blood
  • Actins / metabolism
  • Animals
  • Bone Marrow Cells / cytology
  • Bone Marrow Cells / drug effects
  • Bone Marrow Cells / enzymology
  • Boron Compounds / pharmacology
  • Calcium / blood
  • Calcium / metabolism
  • Calcium Channels / blood
  • Cell Degranulation / drug effects
  • Cell Degranulation / genetics*
  • Cells, Cultured
  • Glucocorticoids / blood
  • Glucocorticoids / physiology*
  • Immediate-Early Proteins / blood
  • Immediate-Early Proteins / deficiency
  • Immediate-Early Proteins / metabolism*
  • Mast Cells / drug effects
  • Mast Cells / enzymology*
  • Mast Cells / metabolism
  • Mice
  • Mice, Knockout
  • Protein Serine-Threonine Kinases / blood
  • Protein Serine-Threonine Kinases / deficiency
  • Protein Serine-Threonine Kinases / metabolism*

Substances

  • Actins
  • Boron Compounds
  • Calcium Channels
  • Glucocorticoids
  • Immediate-Early Proteins
  • 2-aminoethoxydiphenyl borate
  • Protein Serine-Threonine Kinases
  • serum-glucocorticoid regulated kinase
  • Calcium