Mechanisms of itch evoked by β-alanine

J Neurosci. 2012 Oct 17;32(42):14532-7. doi: 10.1523/JNEUROSCI.3509-12.2012.

Abstract

β-Alanine, a popular supplement for muscle building, induces itch and tingling after consumption, but the underlying molecular and neural mechanisms are obscure. Here we show that, in mice, β-alanine elicited itch-associated behavior that requires MrgprD, a G-protein-coupled receptor expressed by a subpopulation of primary sensory neurons. These neurons exclusively innervate the skin, respond to β-alanine, heat, and mechanical noxious stimuli but do not respond to histamine. In humans, intradermally injected β-alanine induced itch but neither wheal nor flare, suggesting that the itch was not mediated by histamine. Thus, the primary sensory neurons responsive to β-alanine are likely part of a histamine-independent itch neural circuit and a target for treating clinical itch that is unrelieved by anti-histamines.

Publication types

  • Research Support, N.I.H., Extramural
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Adult
  • Animals
  • Female
  • Ganglia, Spinal / metabolism
  • Ganglia, Spinal / physiology
  • Gene Knock-In Techniques
  • Humans
  • Injections, Intradermal / methods
  • Male
  • Mice
  • Mice, Inbred C57BL
  • Mice, Knockout
  • Middle Aged
  • Pruritus / etiology*
  • Pruritus / genetics
  • Pruritus / metabolism*
  • Receptors, G-Protein-Coupled / biosynthesis*
  • Receptors, G-Protein-Coupled / deficiency
  • Receptors, G-Protein-Coupled / physiology
  • Sensory Receptor Cells / metabolism
  • Sensory Receptor Cells / pathology
  • Young Adult
  • beta-Alanine / toxicity*

Substances

  • Mrgprd protein, mouse
  • Receptors, G-Protein-Coupled
  • beta-Alanine