Androgen receptors--a method to measure functional behaviour in human prostatic cancer

Eur Urol. 1990;17(1):66-8. doi: 10.1159/000464003.

Abstract

Androgen receptors were measured in soluble and nuclear fractions of tissues obtained from 25 patients. A method using mibolerone, a synthetic androgen, as a ligand is described. This method, which includes the presence of excess ORG 2058 to eliminate interaction with progesterone receptors, gives a reliable determination of androgen receptor content and has been used to predict response to hormonal treatment. However, the results suggest that the presence of functional receptor is not, in itself, a sufficient index of hormonal dependence of the tumour.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Aged
  • Aged, 80 and over
  • Diethylstilbestrol / therapeutic use
  • Humans
  • Male
  • Middle Aged
  • Orchiectomy
  • Prostatic Neoplasms / analysis*
  • Prostatic Neoplasms / drug therapy
  • Prostatic Neoplasms / surgery
  • Receptors, Androgen / analysis*

Substances

  • Receptors, Androgen
  • Diethylstilbestrol