miR-186 downregulation correlates with poor survival in lung adenocarcinoma, where it interferes with cell-cycle regulation

Cancer Res. 2013 Jan 15;73(2):756-66. doi: 10.1158/0008-5472.CAN-12-2651. Epub 2012 Nov 29.

Abstract

Deeper mechanistic understanding of lung adenocarcinoma (non-small cell lung carcinoma, or NSCLC), a leading cause of cancer-related deaths overall, may lead to more effective therapeutic strategies. In analyzing NSCLC clinical specimens and cell lines, we discovered a uniform decrease in miR-186 (MIR186) expression in comparison with normal lung tissue or epithelial cell lines. miR-186 expression correlated with patient survival, with median overall survival time of 63.0 or 21.5 months in cases exhibiting high or low levels of miR-186, respectively. Enforced overexpression of miR-186 in NSCLC cells inhibited proliferation by inducing G(1)-S checkpoint arrest. Conversely, RNA interference-mediated silencing miR-186 expression promoted cell-cycle progression and accelerated the proliferation of NSCLC cells. Cyclin D1 (CCND1), cyclin-dependent kinase (CDK)2, and CDK6 were each directly targeted for inhibition by miR-186 and restoring their expression reversed miR-186-mediated inhibition of cell-cycle progression. The inverse relationship between expression of miR-186 and its targets was confirmed in NSCLC tumor xenografts and clinical specimens. Taken together, our findings established a tumor-suppressive role for miR-186 in the progression of NSCLC.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Adenocarcinoma / genetics*
  • Adenocarcinoma / mortality
  • Adenocarcinoma of Lung
  • Cell Cycle
  • Cell Cycle Checkpoints
  • Cell Line, Tumor
  • Cell Proliferation
  • Cyclin D1 / metabolism
  • Cyclin D2 / metabolism
  • Cyclin-Dependent Kinase 6 / metabolism
  • Down-Regulation*
  • Gene Expression Regulation, Neoplastic*
  • Humans
  • Lung Neoplasms / genetics*
  • Lung Neoplasms / mortality
  • MicroRNAs / metabolism*
  • RNA, Small Interfering / pharmacology

Substances

  • CCND2 protein, human
  • Cyclin D2
  • MIRN1186 microRNA, mouse
  • MicroRNAs
  • RNA, Small Interfering
  • Cyclin D1
  • Cyclin-Dependent Kinase 6