Spectroscopic study on the interaction of catalase with bifendate and analogs

Spectrochim Acta A Mol Biomol Spectrosc. 2013 Feb:102:88-98. doi: 10.1016/j.saa.2012.10.039. Epub 2012 Nov 1.

Abstract

The interactions of bifendate (DDB) or analogs (Bicyclol, I, II and III) with catalase are analyzed by spectrophotometric methods. The fluorescence spectra results show the intrinsic fluorescence of catalase is strongly quenched by DDB or analogs with a static quenching procedure. The binding constants are obtained at three temperatures. The thermodynamics parameters (ΔH, ΔS, ΔG) indicate the hydrophobic and electrostatic interactions play a major role in the interaction. The results of synchronous fluorescence, UV-vis absorption and three-dimensional fluorescence spectra demonstrate that the microenvironments of Trp residue of catalase are disturbed by the analogs. Thermodynamic results showed that DDB is the strongest quencher and bind to catalase with the highest affinity among five compounds.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Antiviral Agents / chemistry
  • Antiviral Agents / pharmacology*
  • Binding Sites
  • Biphenyl Compounds / chemistry
  • Biphenyl Compounds / pharmacology*
  • Catalase / metabolism*
  • Cattle
  • Hepatitis / drug therapy
  • Liver / enzymology*
  • Spectrometry, Fluorescence
  • Thermodynamics

Substances

  • Antiviral Agents
  • Biphenyl Compounds
  • bifendate
  • bicyclol
  • Catalase