Histone demethylase Jumonji D3 (JMJD3) as a tumor suppressor by regulating p53 protein nuclear stabilization

PLoS One. 2012;7(12):e51407. doi: 10.1371/journal.pone.0051407. Epub 2012 Dec 7.

Abstract

Histone methylation regulates normal stem cell fate decisions through a coordinated interplay between histone methyltransferases and demethylases at lineage specific genes. Malignant transformation is associated with aberrant accumulation of repressive histone modifications, such as polycomb mediated histone 3 lysine 27 (H3K27me3) resulting in a histone methylation mediated block to differentiation. The relevance, however, of histone demethylases in cancer remains less clear. We report that JMJD3, a H3K27me3 demethylase, is induced during differentiation of glioblastoma stem cells (GSCs), where it promotes a differentiation-like phenotype via chromatin dependent (INK4A/ARF locus activation) and chromatin independent (nuclear p53 protein stabilization) mechanisms. Our findings indicate that deregulation of JMJD3 may contribute to gliomagenesis via inhibition of the p53 pathway resulting in a block to terminal differentiation.

Publication types

  • Research Support, N.I.H., Extramural
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Blotting, Western
  • Cell Differentiation / physiology*
  • Cell Transformation, Neoplastic / metabolism*
  • DNA Primers / genetics
  • Glioblastoma / physiopathology*
  • Histones / metabolism
  • Humans
  • Immunohistochemistry
  • Immunoprecipitation
  • Jumonji Domain-Containing Histone Demethylases / metabolism*
  • Luciferases
  • Mass Spectrometry
  • Mice
  • Mice, SCID
  • Neoplastic Stem Cells / physiology*
  • Protein Stability
  • Real-Time Polymerase Chain Reaction
  • Tumor Suppressor Protein p53 / metabolism*

Substances

  • DNA Primers
  • Histones
  • Tumor Suppressor Protein p53
  • Luciferases
  • Jumonji Domain-Containing Histone Demethylases
  • KDM6B protein, human