Identification of acidic heterocycle-substituted 1H-pyrazolo[3,4-b]pyridines as soluble guanylate cyclase stimulators

Bioorg Med Chem Lett. 2013 Mar 1;23(5):1197-200. doi: 10.1016/j.bmcl.2013.01.028. Epub 2013 Jan 16.

Abstract

Novel guanylate cyclase stimulators are disclosed. Design, synthesis, SAR, and pharmacological profile of the compounds are discussed.

MeSH terms

  • Animals
  • Guanylate Cyclase / chemistry
  • Guanylate Cyclase / metabolism*
  • Pyrazoles / chemical synthesis
  • Pyrazoles / chemistry*
  • Pyrazoles / pharmacology*
  • Pyridines / chemical synthesis
  • Pyridines / chemistry*
  • Pyridines / pharmacology*
  • Rats
  • Stimulation, Chemical
  • Structure-Activity Relationship

Substances

  • Pyrazoles
  • Pyridines
  • Guanylate Cyclase