A new antiarrhythmic drug in the treatment of recent-onset atrial fibrillation: vernakalant

Cardiovasc Ther. 2013 Oct;31(5):e55-62. doi: 10.1111/1755-5922.12026.

Abstract

Vernakalant is a new antiarrhythmic agent recently approved in Europe for the rapid cardioversion of recent-onset atrial fibrillation. It works by blocking early-activating K+ atrial channels and frequency-dependent atrial Na+ channels, prolonging atrial refractory periods and rate-dependent slowing atrial conduction, without promoting ventricular arrhythmia. Preclinical and clinical trials showed good toleration of this drug. The main purpose of our review is to describe all the trials that led to the incorporation of vernakalant into the current European atrial fibrillation guidelines.

Keywords: Atrial fibrillation; Cardioversion; Vernakalant.

Publication types

  • Review

MeSH terms

  • Administration, Oral
  • Anisoles / adverse effects
  • Anisoles / chemistry
  • Anisoles / pharmacology
  • Anisoles / therapeutic use*
  • Anti-Arrhythmia Agents / therapeutic use*
  • Atrial Fibrillation / drug therapy*
  • Clinical Trials as Topic
  • Humans
  • Pyrrolidines / adverse effects
  • Pyrrolidines / chemistry
  • Pyrrolidines / pharmacology
  • Pyrrolidines / therapeutic use*

Substances

  • Anisoles
  • Anti-Arrhythmia Agents
  • Pyrrolidines
  • vernakalant