Identification of a calmodulin-binding domain in Sema4D that regulates its exodomain shedding in platelets

Blood. 2013 May 16;121(20):4221-30. doi: 10.1182/blood-2012-11-470609. Epub 2013 Apr 5.

Abstract

Semaphorin 4D (Sema4D) is a transmembrane protein that supports contact-dependent amplification of platelet activation by collagen before being gradually cleaved by the metalloprotease ADAM17, as we have previously shown. Cleavage releases a soluble 120-kDa exodomain fragment for which receptors exist on platelets and endothelial cells. Here we have examined the mechanism that regulates Sema4D exodomain cleavage. The results show that the membrane-proximal cytoplasmic domain of Sema4D contains a binding site for calmodulin within the polybasic region Arg762-Lys779. Coprecipitation studies show that Sema4D and calmodulin are associated in resting platelets, forming a complex that dissociates upon platelet activation by the agonists that trigger Sema4D cleavage. Inhibiting calmodulin with W7 or introducing a membrane-permeable peptide corresponding to the calmodulin-binding site is sufficient to trigger the dissociation of Sema4D from calmodulin and initiate cleavage. Conversely, deletion of the calmodulin-binding site causes constitutive shedding of Sema4D. These results show that (1) Sema4D is a calmodulin-binding protein with a site of interaction in its membrane-proximal cytoplasmic domain, (2) platelet agonists cause dissociation of the calmodulin-Sema4D complex, and (3) dissociation of the complex is sufficient to trigger ADAM17-dependent cleavage of Sema4D, releasing a bioactive fragment.

Publication types

  • Research Support, N.I.H., Extramural
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Amino Acid Sequence
  • Animals
  • Antigens, CD / chemistry*
  • Antigens, CD / genetics
  • Antigens, CD / metabolism*
  • Blood Platelets / drug effects
  • Blood Platelets / metabolism*
  • Blood Platelets / physiology
  • CHO Cells
  • Calmodulin / antagonists & inhibitors
  • Calmodulin / metabolism*
  • Cricetinae
  • Cricetulus
  • Enzyme Inhibitors / pharmacology
  • Humans
  • Molecular Sequence Data
  • Platelet Activation / drug effects
  • Platelet Activation / genetics
  • Protein Binding / drug effects
  • Protein Interaction Domains and Motifs / physiology*
  • Protein Processing, Post-Translational / drug effects
  • Semaphorins / chemistry*
  • Semaphorins / genetics
  • Semaphorins / metabolism*
  • Sulfonamides / pharmacology

Substances

  • Antigens, CD
  • CD100 antigen
  • Calmodulin
  • Enzyme Inhibitors
  • Semaphorins
  • Sulfonamides
  • W 7