Isoflurane and sevoflurane increase interleukin-6 levels through the nuclear factor-kappa B pathway in neuroglioma cells

Br J Anaesth. 2013 Jun;110 Suppl 1(Suppl 1):i82-91. doi: 10.1093/bja/aet115. Epub 2013 Apr 19.

Abstract

Background: Isoflurane can increase pro-inflammatory cytokine interleukin (IL)-6 levels. However, the up-stream mechanism remains unknown. Nuclear factor-kappa B (NF-κB) promotes the generation of pro-inflammatory cytokines. We examined the effects of isoflurane and sevoflurane on the NF-κB signalling pathway and its association with IL-6 levels in cultured cells.

Methods: H4 human neuroglioma cells (H4 cells), and mouse primary neurones and microglia were treated with 2% isoflurane or 4.1% sevoflurane for 6 h, for analysis of IL-6 and NF-κB. Pyrrolidine dithiocarbamate (an NF-κB inhibitor) or 2-deoxy-d-glucose (2-DG) (an inhibitor of glucose glycolysis) was applied 1 h before anaesthetic treatment.

Results: Isoflurane or sevoflurane treatment increased the levels of IL-6 [isoflurane: 410% (54); sevoflurane: 290% (24)], the nuclear levels of NF-κB [isoflurane: 170% (36); sevoflurane: 320% (30)], and the transcription activity of NF-κB in H4 cells. Moreover, isoflurane enhanced the transcription activity of NF-κB in mouse microglia, but not primary neurones. Finally, pyrrolidine dithiocarbamate and 2-DG attenuated isoflurane-induced increases in IL-6 and NF-κB, and the transcription activity of NF-κB.

Conclusions: These studies in H4 cells suggest that the NF-κB signalling pathway could contribute to isoflurane or sevoflurane-induced neuroinflammation. This could lead to the targeted intervention of anaesthetic-induced neuroinflammation.

Keywords: NF-κB; anaesthetic; interleukin-6.

Publication types

  • Research Support, N.I.H., Extramural
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Anesthetics, Inhalation / antagonists & inhibitors
  • Anesthetics, Inhalation / pharmacology*
  • Animals
  • Antimetabolites / pharmacology
  • Cell Nucleus / metabolism
  • Cells, Cultured
  • Deoxyglucose / pharmacology
  • Glioma
  • Humans
  • Inflammation Mediators / metabolism*
  • Interleukin-6 / biosynthesis*
  • Isoflurane / antagonists & inhibitors
  • Isoflurane / pharmacology
  • Methyl Ethers / pharmacology
  • Mice
  • Microglia / drug effects*
  • Microglia / metabolism
  • NF-kappa B / antagonists & inhibitors
  • NF-kappa B / biosynthesis
  • NF-kappa B / physiology*
  • Neurons / drug effects*
  • Neurons / metabolism
  • Proline / analogs & derivatives
  • Proline / pharmacology
  • Sevoflurane
  • Signal Transduction / drug effects
  • Signal Transduction / physiology
  • Thiocarbamates / pharmacology
  • Transcription, Genetic / drug effects
  • Tumor Cells, Cultured

Substances

  • Anesthetics, Inhalation
  • Antimetabolites
  • Inflammation Mediators
  • Interleukin-6
  • Methyl Ethers
  • NF-kappa B
  • Thiocarbamates
  • prolinedithiocarbamate
  • Sevoflurane
  • Proline
  • Deoxyglucose
  • Isoflurane