Growth hormone potentiates 17β-estradiol-dependent breast cancer cell proliferation independently of IGF-I receptor signaling

Endocrinology. 2013 Sep;154(9):3219-27. doi: 10.1210/en.2012-2208. Epub 2013 Jun 19.

Abstract

Estrogen action in mammary gland development and breast cancer progression is tightly linked to the GH/IGF-I axis. Although many of the effects of GH on mammary gland growth and development require IGF-I, the extent to which GH action in breast cancer depends on IGF-I is not known. We examined GH action in a panel of estrogen receptor-positive breast cancer cell lines and found that T47D cells express significant levels of GH receptor and that GH significantly enhances 17β-estradiol (E2)-stimulated proliferation in these cells. GH action in the T47D cells was independent of changes in IGF-I and IGF-I receptor (IGF-IR) expression and IGF-IR signaling, suggesting that GH can exert direct effects on breast cancer cells. Although E2-dependent proliferation required IGF-IR signaling, the combination of GH+E2 overcame inhibition of IGF-IR activity to restore proliferation. In contrast, GH required both Janus kinase 2 and epidermal growth factor receptor signaling for subsequent ERK activation and potentiation of E2-dependent proliferation. Downstream of these pathways, we identified a number of immediate early-response genes associated with proliferation that are rapidly and robustly up-regulated by GH. These findings demonstrate that GH can have important effects in breast cancer cells that are distinct from IGF-IR activity, suggesting that novel drugs or improved combination therapies targeting estrogen receptor and the GH/IGF axis may be beneficial for breast cancer patients.

Publication types

  • Comparative Study
  • Research Support, N.I.H., Extramural
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Antineoplastic Agents / pharmacology
  • Breast Neoplasms / drug therapy
  • Breast Neoplasms / metabolism*
  • Cell Line, Tumor
  • Cell Proliferation / drug effects
  • ErbB Receptors / genetics
  • ErbB Receptors / metabolism
  • Estradiol / metabolism*
  • Female
  • Human Growth Hormone / genetics
  • Human Growth Hormone / metabolism*
  • Humans
  • Insulin-Like Growth Factor I / antagonists & inhibitors
  • Insulin-Like Growth Factor I / genetics
  • Insulin-Like Growth Factor I / metabolism*
  • Janus Kinase 2 / genetics
  • Janus Kinase 2 / metabolism
  • MAP Kinase Signaling System / drug effects
  • Neoplasm Proteins / antagonists & inhibitors
  • Neoplasm Proteins / genetics
  • Neoplasm Proteins / metabolism
  • Protein Kinase Inhibitors / pharmacology
  • RNA, Messenger / metabolism
  • Receptor, IGF Type 1 / antagonists & inhibitors
  • Receptor, IGF Type 1 / genetics
  • Receptor, IGF Type 1 / metabolism*
  • Receptors, Somatotropin / genetics
  • Receptors, Somatotropin / metabolism*
  • Recombinant Proteins / metabolism
  • Signal Transduction* / drug effects
  • Up-Regulation / drug effects

Substances

  • Antineoplastic Agents
  • IGF1 protein, human
  • Neoplasm Proteins
  • Protein Kinase Inhibitors
  • RNA, Messenger
  • Receptors, Somatotropin
  • Recombinant Proteins
  • Human Growth Hormone
  • Estradiol
  • Insulin-Like Growth Factor I
  • EGFR protein, human
  • ErbB Receptors
  • Receptor, IGF Type 1
  • JAK2 protein, human
  • Janus Kinase 2