Optimising measles virus-guided radiovirotherapy with external beam radiotherapy and specific checkpoint kinase 1 inhibition

Radiother Oncol. 2013 Jul;108(1):24-31. doi: 10.1016/j.radonc.2013.05.036. Epub 2013 Jul 9.

Abstract

Background and purpose: We previously reported a therapeutic strategy comprising replication-defective NIS-expressing adenovirus combined with radioiodide, external beam radiotherapy (EBRT) and DNA repair inhibition. We have now evaluated NIS-expressing oncolytic measles virus (MV-NIS) combined with NIS-guided radioiodide, EBRT and specific checkpoint kinase 1 (Chk1) inhibition in head and neck and colorectal models.

Materials and methods: Anti-proliferative/cytotoxic effects of individual agents and their combinations were measured by MTS, clonogenic and Western analysis. Viral gene expression was measured by radioisotope uptake and replication by one-step growth curves. Potential synergistic interactions were tested in vitro by Bliss independence analysis and in in vivo therapeutic studies.

Results: EBRT and MV-NIS were synergistic in vitro. Furthermore, EBRT increased NIS expression in infected cells. SAR-020106 was synergistic with EBRT, but also with MV-NIS in HN5 cells. MV-NIS mediated (131)I-induced cytotoxicity in HN5 and HCT116 cells and, in the latter, this was enhanced by SAR-020106. In vivo studies confirmed that MV-NIS, EBRT and Chk1 inhibition were effective in HCT116 xenografts. The quadruplet regimen of MV-NIS, virally-directed (131)I, EBRT and SAR-020106 had significant anti-tumour activity in HCT116 xenografts.

Conclusion: This study strongly supports translational and clinical research on MV-NIS combined with radiation therapy and radiosensitising agents.

Keywords: External beam radiation therapy; Oncolytic measles virus; Radiation-sensitizing agents; Radiovirotherapy.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Cell Line, Tumor
  • Checkpoint Kinase 1
  • Colorectal Neoplasms / therapy*
  • Combined Modality Therapy
  • Head and Neck Neoplasms / therapy*
  • Humans
  • Iodine Radioisotopes / therapeutic use*
  • Isoquinolines / therapeutic use*
  • Measles virus / physiology*
  • Mice
  • Oncolytic Virotherapy*
  • Protein Kinase Inhibitors / therapeutic use*
  • Protein Kinases / physiology*
  • Pyrazines / therapeutic use*
  • Radiation-Sensitizing Agents / therapeutic use*
  • Symporters / genetics
  • Virus Replication
  • Xenograft Model Antitumor Assays

Substances

  • Iodine Radioisotopes
  • Isoquinolines
  • Protein Kinase Inhibitors
  • Pyrazines
  • Radiation-Sensitizing Agents
  • SAR 020106
  • Symporters
  • sodium-iodide symporter
  • Protein Kinases
  • CHEK1 protein, human
  • Checkpoint Kinase 1
  • Chek1 protein, mouse