The effects of congenital brain serotonin deficiency on responses to chronic fluoxetine

Transl Psychiatry. 2013 Aug 13;3(8):e291. doi: 10.1038/tp.2013.65.

Abstract

The importance of reversing brain serotonin (5-HT) deficiency and promoting hippocampal neurogenesis in the mechanisms of action for antidepressants remain highly controversial. Here we examined the behavioral, neurochemical and neurogenic effects of chronic fluoxetine (FLX) in a mouse model of congenital 5-HT deficiency, the tryptophan hydroxylase 2 (R439H) knock-in (Tph2KI) mouse. Our results demonstrate that congenital 5-HT deficiency prevents a subset of the signature molecular, cellular and behavioral effects of FLX, despite the fact that FLX restores the 5-HT levels of Tph2KI mice to essentially the levels observed in wild-type mice at baseline. These results suggest that inducing supra-physiological levels of 5-HT, not merely reversing 5-HT deficiency, is required for many of the antidepressant-like effects of FLX. We also demonstrate that co-administration of the 5-HT precursor, 5-hydroxytryptophan (5-HTP), along with FLX rescues the novelty suppressed feeding (NSF) anxiolytic-like effect of FLX in Tph2KI mice, despite still failing to induce neurogenesis. Thus, our results indicate that brain 5-HT deficiency reduces the efficacy of FLX and that supplementation with 5-HTP can restore some antidepressant-like responses in the context of 5-HT deficiency. Our findings also suggest that feeding latency reductions in the NSF induced by chronic 5-HT elevation are not mediated by drug-induced increments in neurogenesis in 5-HT-deficient animals. Overall, these findings shed new light on the impact of 5-HT deficiency on responses to FLX and may have important implications for treatment selection in depression and anxiety disorders.

Publication types

  • Research Support, N.I.H., Extramural
  • Research Support, Non-U.S. Gov't

MeSH terms

  • 5-Hydroxytryptophan / pharmacology
  • Animals
  • Antidepressive Agents, Second-Generation / pharmacology
  • Anxiety / metabolism
  • Behavior, Animal / drug effects*
  • Feeding Behavior / drug effects
  • Fluoxetine / pharmacology*
  • Hippocampus / drug effects*
  • Hippocampus / metabolism
  • Mice
  • Mice, Transgenic
  • Microdialysis
  • Neurogenesis / drug effects*
  • Selective Serotonin Reuptake Inhibitors / pharmacology*
  • Serotonin / deficiency*
  • Serotonin / metabolism
  • Tryptophan Hydroxylase / genetics

Substances

  • Antidepressive Agents, Second-Generation
  • Serotonin Uptake Inhibitors
  • Fluoxetine
  • Serotonin
  • 5-Hydroxytryptophan
  • Tph2 protein, mouse
  • Tryptophan Hydroxylase