Somatic and psychological effects of low-dose aromatase inhibition in men with obesity-related hypogonadotropic hypotestosteronemia

Eur J Endocrinol. 2013 Oct 8;169(5):705-14. doi: 10.1530/EJE-13-0190. Print 2013 Nov.

Abstract

Introduction: Reduced testosterone levels are frequently observed in obese men. Increased aromatase activity may be an etiological factor.

Objective: In this study, we evaluate the clinical effects of aromatase inhibition in obesity-related hypogonadotropic hypotestosteronemia (OrHH).

Methods: Double-blind, placebo-controlled, 6-month trial in 42 obese men with a BMI >35 kg/m(2), and a serum total testosterone <10 nmol/l. All patients started on one tablet of 2.5 mg/week, with subsequent dose escalation every month until a serum total testosterone of 20 nmol/l was reached.

Endpoints: Psychological function, body composition, exercise capacity, and glucose, lipid, and bone metabolism.

Results: Thirty-nine patients completed the study according to protocol. Letrozole decreased serum estradiol from 119.1±10.1 to 59.2±6.1 pmol/l (P<0.001), and increased serum LH from 3.3±0.3 to 8.8±0.9 U/l (P<0.0001) and serum total testosterone from 8.6±0.7 to 21.5±1.3 nmol/l (P<0.0001). Significant effects on the predefined endpoints were not observed.

Conclusion: Despite a marked rise in serum testosterone, low-dose aromatase inhibition had no somatic or psychological effects in men with OrHH.

Publication types

  • Randomized Controlled Trial

MeSH terms

  • Adult
  • Androgens / blood
  • Aromatase Inhibitors / administration & dosage
  • Aromatase Inhibitors / adverse effects
  • Aromatase Inhibitors / therapeutic use*
  • Blood Glucose / metabolism
  • Body Composition / drug effects
  • Body Mass Index
  • Bone Density / drug effects
  • Double-Blind Method
  • Energy Intake
  • Estradiol / blood
  • Exercise Tolerance / drug effects
  • Exercise Tolerance / physiology
  • Hormones / blood
  • Humans
  • Hypogonadism / blood*
  • Hypogonadism / complications*
  • Hypogonadism / psychology
  • Letrozole
  • Lipid Metabolism / drug effects
  • Luteinizing Hormone / blood
  • Male
  • Middle Aged
  • Neuropsychological Tests
  • Nitriles / administration & dosage
  • Nitriles / adverse effects
  • Nitriles / therapeutic use*
  • Obesity, Morbid / blood*
  • Obesity, Morbid / complications*
  • Obesity, Morbid / psychology
  • Psychometrics
  • Testosterone / blood
  • Testosterone / deficiency*
  • Triazoles / administration & dosage
  • Triazoles / adverse effects
  • Triazoles / therapeutic use*

Substances

  • Androgens
  • Aromatase Inhibitors
  • Blood Glucose
  • Hormones
  • Nitriles
  • Triazoles
  • Testosterone
  • Estradiol
  • Letrozole
  • Luteinizing Hormone