[Ruxolitinib prescription in myelofibrosis]

Bull Cancer. 2013 Sep;100(9):897-902. doi: 10.1684/bdc.2013.1792.
[Article in French]

Abstract

Ruxolitinib is a JAK/STAT inhibitor, which has demonstrated clinical benefits in patients with intermediate-2 and high-risk myelofibrosis. Moreover, first results of recent clinical trials show a trend to better overall survival with ruxolitinib, which allows to hope that we will soon be able to change the natural evolution of this poor outcome disease. With such results, ruxolitinib quickly obtained the Food and Drug Administration (FDA) approval in the United States of America. In France, ruxolitinib is now available, allowing its administration to symptomatic myelofibrosis patients.

Keywords: myeloproliferative syndrome; primary myelofibrosis; ruxolitinib; splenomegaly.

Publication types

  • Review

MeSH terms

  • Drug Interactions
  • Humans
  • Janus Kinase 1 / genetics
  • Janus Kinase 2 / genetics
  • Janus Kinases / antagonists & inhibitors*
  • Janus Kinases / physiology
  • Myeloproliferative Disorders / drug therapy
  • Myeloproliferative Disorders / genetics
  • Nitriles
  • Philadelphia Chromosome
  • Primary Myelofibrosis / drug therapy*
  • Primary Myelofibrosis / mortality
  • Prognosis
  • Pyrazoles / adverse effects
  • Pyrazoles / pharmacokinetics
  • Pyrazoles / therapeutic use*
  • Pyrimidines
  • Remission Induction
  • Splenomegaly / drug therapy

Substances

  • Nitriles
  • Pyrazoles
  • Pyrimidines
  • ruxolitinib
  • Janus Kinase 1
  • Janus Kinase 2
  • Janus Kinases