Ginsenoside Rb1 protects rat retinal ganglion cells against hypoxia and oxidative stress

Mol Med Rep. 2013 Nov;8(5):1397-403. doi: 10.3892/mmr.2013.1658. Epub 2013 Aug 28.

Abstract

The current study was designed to investigate the effect of ginsenoside Rb1 (Rb1) on apoptosis induced by hypoxia and oxidative stress in a retinal ganglion cell line (RGC-5). The underlying mechanism was also investigated. RGC-5 cells were pretreated with 10 µmol/l Rb1 for 24 h and exposed to 400 µmol/l cobalt chloride (CoCl2) for 48 h or 600 µmol/l H2O2 for 24 h. The percentage of cells actively undergoing apoptosis was determined by flow cytometry with Annexin V/propidium iodide (PI) double staining. The expression of caspases was determined using western blot analysis. CoCl2 and H2O2 treatments significantly increased the apoptotic percentages to 24.5 and 21.63%, respectively. Pretreatment of Rb1 reduced the total apoptotic percentages to 15.12 and 12.03%, respectively. The expression of cleaved caspase-3, -9 and -8 was increased in the CoCl2-treated group, however, caspase-3 was not increased in the H2O2-treated group. Pretreatment of Rb1 reduced the expression of cleaved caspase-3 and -9 in the CoCl2-treated group, but reduced only cleaved caspase-9 in the H2O2-treated group. These results suggest that Rb1 may prevent RGC-5 cells from apoptosis against hypoxia and oxidative stress via the mitochondrial pathway.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Antimutagenic Agents / pharmacology
  • Apoptosis / drug effects
  • Blotting, Western
  • Cell Proliferation / drug effects
  • Cells, Cultured
  • Cobalt / pharmacology
  • Ginsenosides / pharmacology*
  • Hydrogen Peroxide / pharmacology
  • Hypoxia / drug therapy*
  • Hypoxia / metabolism
  • Hypoxia / pathology
  • Neuroprotective Agents / pharmacology*
  • Oxidants / pharmacology
  • Oxidative Stress / drug effects*
  • RNA, Messenger
  • Rats
  • Rats, Sprague-Dawley
  • Retinal Ganglion Cells / cytology
  • Retinal Ganglion Cells / drug effects*
  • Retinal Ganglion Cells / metabolism

Substances

  • Antimutagenic Agents
  • Ginsenosides
  • Neuroprotective Agents
  • Oxidants
  • RNA, Messenger
  • Cobalt
  • ginsenoside Rb1
  • Hydrogen Peroxide
  • cobaltous chloride