Abstract
A direct switch of candesartan to the fixed-dose combination olmesartan/amlodipine in uncontrolled hypertension is a frequent clinical requirement but is not covered by current labeling. An open-label, prospective, single-arm phase IIIb study was performed in patients with 32 mg candesartan followed by olmesartan/amlodipine 40/10 mg. The primary endpoint was change in mean daytime systolic blood pressure (BP). Mean daytime systolic BP was reduced by 9.2±12.6 mm Hg (P<.0001) after substituting candesartan for olmesartan/amlodipine (baseline BP 140.2±9.7 mm Hg). The reduction in office BP was 9.4±18.4/4.0±9.6 mm Hg; P<.002). Overall, 61.3% of patients achieved a target BP <140/90 mm Hg using office BP and <135/85 mm Hg using ambulatory BP measurement. There were 8 adverse events with a possible relation to study drug and 1 unrelated serious adverse events. In conclusion, patients with uncontrolled moderate arterial hypertension being treated using candesartan monotherapy achieve a further reduction of BP when switched directly to a fixed-dose combination of olmesartan 40 mg/amlodipine 10 mg.
©2013 Wiley Periodicals, Inc.
Publication types
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Clinical Trial, Phase III
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Multicenter Study
MeSH terms
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Aged
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Amlodipine / administration & dosage
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Amlodipine / pharmacology
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Amlodipine / therapeutic use*
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Angiotensin Receptor Antagonists / administration & dosage
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Angiotensin Receptor Antagonists / pharmacology
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Angiotensin Receptor Antagonists / therapeutic use*
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Antihypertensive Agents / administration & dosage
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Antihypertensive Agents / pharmacology
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Antihypertensive Agents / therapeutic use
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Benzimidazoles / administration & dosage
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Benzimidazoles / pharmacology
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Benzimidazoles / therapeutic use*
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Biphenyl Compounds
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Blood Pressure / drug effects
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Blood Pressure / physiology*
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Calcium Channel Blockers / administration & dosage
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Calcium Channel Blockers / pharmacology
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Calcium Channel Blockers / therapeutic use*
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Circadian Rhythm / physiology
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Dose-Response Relationship, Drug
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Drug Administration Schedule
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Drug Therapy, Combination
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Essential Hypertension
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Female
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Humans
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Hypertension / drug therapy*
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Hypertension / physiopathology
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Imidazoles / administration & dosage
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Imidazoles / pharmacology
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Imidazoles / therapeutic use*
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Male
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Middle Aged
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Prospective Studies
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Systole / drug effects
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Systole / physiology
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Tetrazoles / administration & dosage
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Tetrazoles / pharmacology
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Tetrazoles / therapeutic use*
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Treatment Outcome
Substances
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Angiotensin Receptor Antagonists
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Antihypertensive Agents
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Benzimidazoles
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Biphenyl Compounds
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Calcium Channel Blockers
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Imidazoles
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Tetrazoles
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Amlodipine
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olmesartan
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candesartan