Genetic ablation of 12/15-lipoxygenase but not 5-lipoxygenase protects against denervation-induced muscle atrophy

Free Radic Biol Med. 2014 Feb:67:30-40. doi: 10.1016/j.freeradbiomed.2013.10.002. Epub 2013 Oct 8.

Abstract

Skeletal muscle atrophy is a debilitating outcome of a number of chronic diseases and conditions associated with loss of muscle innervation by motor neurons, such as aging and neurodegenerative diseases. We previously reported that denervation-induced loss of muscle mass is associated with activation of cytosolic phospholipase A2 (cPLA2), the rate-limiting step for the release of arachidonic acid from membrane phospholipids, which then acts as a substrate for metabolic pathways that generate bioactive lipid mediators. In this study, we asked whether 5- and 12/15-lipoxygenase (LO) lipid metabolic pathways downstream of cPLA2 mediate denervation-induced muscle atrophy in mice. Both 5- and 12/15-LO were activated in response to surgical denervation; however, 12/15-LO activity was increased ~2.5-fold versus an ~1.5-fold increase in activity of 5-LO. Genetic and pharmacological inhibition of 12/15-LO (but not 5-LO) significantly protected against denervation-induced muscle atrophy, suggesting a selective role for the 12/15-LO pathway in neurogenic muscle atrophy. The activation of the 12/15-LO pathway (but not 5-LO) during muscle atrophy increased NADPH oxidase activity, protein ubiquitination, and ubiquitin-proteasome-mediated proteolytic degradation. In conclusion, this study reveals a novel pathway for neurogenic muscle atrophy and suggests that 12/15-LO may be a potential therapeutic target in diseases associated with loss of innervation and muscle atrophy.

Keywords: 12/15-Lipoxygenase; 5-Lipoxygenase; Denervation; Free radicals; Muscle atrophy; NADPH oxidase.

Publication types

  • Research Support, N.I.H., Extramural

MeSH terms

  • Animals
  • Arachidonate 12-Lipoxygenase / deficiency*
  • Arachidonate 12-Lipoxygenase / genetics
  • Arachidonate 15-Lipoxygenase / deficiency*
  • Arachidonate 15-Lipoxygenase / genetics
  • Arachidonate 5-Lipoxygenase / deficiency*
  • Arachidonate 5-Lipoxygenase / genetics
  • Enzyme Inhibitors / pharmacology
  • Flavanones / pharmacology
  • Fluorenes / pharmacology
  • Gene Deletion*
  • Gene Expression
  • Genetic Therapy
  • Male
  • Mice
  • Mice, Knockout
  • Muscle Denervation
  • Muscle, Skeletal / enzymology*
  • Muscle, Skeletal / innervation
  • Muscle, Skeletal / physiopathology
  • Muscle, Skeletal / surgery
  • Muscular Atrophy / enzymology
  • Muscular Atrophy / genetics*
  • Muscular Atrophy / physiopathology
  • Muscular Atrophy / therapy*
  • NADPH Oxidases / genetics
  • NADPH Oxidases / metabolism
  • Proteasome Endopeptidase Complex / metabolism
  • Proteolysis / drug effects
  • Signal Transduction
  • Ubiquitination / drug effects

Substances

  • 12-15-lipoxygenase
  • 6,11-dihydro-5-thia-11-aza-benzo(a)-fluorene
  • Enzyme Inhibitors
  • Flavanones
  • Fluorenes
  • baicalein
  • Arachidonate 12-Lipoxygenase
  • Arachidonate 15-Lipoxygenase
  • Arachidonate 5-Lipoxygenase
  • NADPH Oxidases
  • Proteasome Endopeptidase Complex