Folic acid conjugated self-assembled layered double hydroxide nanoparticles for high-efficacy-targeted drug delivery

Chem Commun (Camb). 2013 Dec 4;49(93):10938-40. doi: 10.1039/c3cc45714a.

Abstract

Enhanced selectivity and efficacy is important for advanced drug delivery. Herein, a novel type of folic acid conjugated self-assembled layered double hydroxide nanoparticles is reported. These nanoparticles have a drug loading capacity of 27 wt% and are able to enter cell nuclei and dramatically improve the efficacy of MTX.

MeSH terms

  • Cell Line, Tumor
  • Cell Nucleus / chemistry
  • Cell Nucleus / metabolism
  • Cell Survival / drug effects
  • Drug Carriers / chemistry*
  • Folic Acid / chemistry*
  • HeLa Cells
  • Humans
  • Hydroxides / chemistry*
  • Methotrexate / chemistry
  • Methotrexate / toxicity
  • Microscopy, Confocal
  • Nanoparticles / chemistry*

Substances

  • Drug Carriers
  • Hydroxides
  • hydroxide ion
  • Folic Acid
  • Methotrexate