Combination therapy in pulmonary arterial hypertension

Clin Chest Med. 2013 Dec;34(4):841-55. doi: 10.1016/j.ccm.2013.08.007. Epub 2013 Oct 17.

Abstract

Despite major advances in understanding the mechanisms of disease and development of specific drug therapy, pulmonary arterial hypertension (PAH) remains a progressive, fatal disease. At present there are 3 classes of drug therapy for PAH: prostaglandins, endothelin receptor antagonists, and phosphodiesterase-5 inhibitors. To maximize therapeutic benefit, and according to national and international guidelines, many patients are treated with combinations of these medications. This review presents a detailed account of the published data on the use of combination therapy in PAH. There are few randomized, placebo-controlled trial data to strongly support efficacy of most combination therapy, particularly oral combination therapy.

Keywords: Combination therapy; Endothelin receptor antagonists; Phosphodiesterase-5 inhibitors; Prostacyclin; Pulmonary arterial hypertension; Treatment.

Publication types

  • Review

MeSH terms

  • Drug Therapy, Combination
  • Endothelin Receptor Antagonists*
  • Epoprostenol / analogs & derivatives*
  • Epoprostenol / therapeutic use
  • Familial Primary Pulmonary Hypertension
  • Humans
  • Hypertension, Pulmonary / drug therapy*
  • Phosphodiesterase 5 Inhibitors / therapeutic use*
  • Prostaglandins / therapeutic use

Substances

  • Endothelin Receptor Antagonists
  • Phosphodiesterase 5 Inhibitors
  • Prostaglandins
  • Epoprostenol