Etifoxine provides benefits in nerve repair with acellular nerve grafts

Muscle Nerve. 2014 Aug;50(2):235-43. doi: 10.1002/mus.24131. Epub 2014 May 15.

Abstract

Introduction: Acellular nerve grafts are good candidates for nerve repair, but the clinical outcome of grafting is not always satisfactory. We investigated whether etifoxine could enhance nerve regeneration.

Methods: Seventy-two Sprague-Dawley rats were divided into 3 groups: (1) autograft; (2) acellular nerve graft; and (3) acellular nerve graft plus etifoxine. Histological and electrophysiological examinations were performed to evaluate the efficacy of nerve regeneration. Walking-track analysis was used to examine functional recovery. Quantitative polymerase chain reaction was used to evaluate changes in mRNA level.

Results: Etifoxine: (i) increased expression of neurofilaments in regenerated axons; (ii) improved sciatic nerve regeneration measured by histological examination; (iii) increased nerve conduction velocity; (iv) improved walking behavior as measured by footprint analysis; and (v) boosted expression of neurotrophins.

Conclusions: These results show that etifoxine can enhance peripheral nerve regeneration across large nerve gaps repaired by acellular nerve grafts by increasing expression of neurotrophins.

Keywords: TSPO; acellular nerve grafts; etifoxine; nerve regeneration; neurotrophins expression.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Disease Models, Animal
  • Electric Stimulation
  • Evoked Potentials / drug effects
  • Gene Expression / drug effects
  • Gene Expression / physiology
  • Glial Cell Line-Derived Neurotrophic Factor / genetics
  • Glial Cell Line-Derived Neurotrophic Factor / metabolism
  • Locomotion / drug effects
  • Male
  • Nerve Growth Factor / genetics
  • Nerve Growth Factor / metabolism
  • Nerve Regeneration / drug effects*
  • Nerve Regeneration / physiology
  • Neural Conduction / drug effects
  • Neural Conduction / physiology
  • Neurofilament Proteins / metabolism
  • Oxazines / pharmacology
  • Oxazines / therapeutic use*
  • Rats
  • Rats, Sprague-Dawley
  • Recovery of Function
  • Sciatic Neuropathy / drug therapy*
  • Sciatic Neuropathy / surgery*
  • Skin / innervation
  • Transplantation, Autologous / methods*
  • Vascular Endothelial Growth Factor A / genetics
  • Vascular Endothelial Growth Factor A / metabolism

Substances

  • Glial Cell Line-Derived Neurotrophic Factor
  • Neurofilament Proteins
  • Oxazines
  • Vascular Endothelial Growth Factor A
  • neurofilament protein H
  • Nerve Growth Factor
  • etifoxine