Identifying potential therapeutic targets of methicillin-resistant Staphylococcus aureus through in vivo proteomic analysis

J Infect Dis. 2014 May 15;209(10):1533-41. doi: 10.1093/infdis/jit662. Epub 2013 Nov 26.

Abstract

Background: Detailed knowledge on protein repertoire of a pathogen during host infection is needed for both developing a better understanding of the pathogenesis and defining potential therapeutic targets. Such data, however, have been missing for Staphylococcus aureus, a major human pathogen.

Methods: We determined the surface proteome of methicillin-resistant S. aureus (MRSA) clone usa300 derived directly from murine systemic infectiON.

Results: The majority of the in vivo-expressed surface-associated proteins were lipoproteins involved in nutrient acquisition, especially uptake of metal ions. Enzyme-linked immunosorbent assay (ELISA) of convalescent human serum samples revealed that proteins that were highly produced during murine experimental infection were also produced during natural human infection. We found that among the 7 highly abundant lipoproteins only MntC, which is the manganese-binding protein of the MntABC system, was essential for MRSA virulence during murine systemic infection. Moreover, we show that MntA and MntB are equally important for MRSA virulence.

Conclusions: Besides providing experimental evidence that MntABC might be a potential therapeutic target for the development of antibiotics, our in vivo proteomics data will serve as a valuable basis for defining potential antigen combinations for multicomponent vaccines.

Keywords: MRSA; Staphylococcus aureus; bacterial pathogenesis; proteomics; vaccine and antibiotic development.

Publication types

  • Research Support, N.I.H., Extramural
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Anti-Bacterial Agents / pharmacology*
  • Bacterial Proteins / genetics
  • Bacterial Proteins / metabolism*
  • Enzyme-Linked Immunosorbent Assay / methods
  • Gene Expression Regulation, Bacterial / physiology*
  • Humans
  • Kidney / microbiology
  • Lipoproteins / genetics
  • Lipoproteins / metabolism
  • Membrane Proteins / genetics
  • Membrane Proteins / metabolism
  • Methicillin-Resistant Staphylococcus aureus / drug effects*
  • Methicillin-Resistant Staphylococcus aureus / metabolism*
  • Methicillin-Resistant Staphylococcus aureus / pathogenicity
  • Mice
  • Proteomics*
  • Serum / immunology
  • Staphylococcal Infections / immunology
  • Staphylococcal Infections / microbiology
  • Staphylococcal Infections / prevention & control
  • Staphylococcal Vaccines / immunology
  • Virulence

Substances

  • Anti-Bacterial Agents
  • Bacterial Proteins
  • Lipoproteins
  • Membrane Proteins
  • Staphylococcal Vaccines