Modulation of adipose tissue thermogenesis as a method for increasing energy expenditure

Bioorg Med Chem Lett. 2014 Jan 15;24(2):425-9. doi: 10.1016/j.bmcl.2013.12.016. Epub 2013 Dec 10.

Abstract

There is a renewed interest in the role of adipose tissue in energy utilization and thermogenesis and its potential application in the treatment of metabolic disorders such as obesity and diabetes. The last few years have seen the identification of brown adipose tissue capable of metabolic activation in adult humans, the possibility of recruiting 'beige' adipocytes to increase energy expenditure, and the implication of molecules such as FGF21 and irisin in inducing increases in energy expenditure in adipose tissue. The translation of these findings into human trials to deliver safe, efficacious medicines remains a challenge.

Keywords: Beige adipose; Brown adipose tissue; Thermogenesis.

Publication types

  • Review

MeSH terms

  • Adipocytes / drug effects
  • Adipocytes / metabolism*
  • Adipose Tissue / drug effects
  • Adipose Tissue / metabolism*
  • Adipose Tissue, Brown / drug effects
  • Adipose Tissue, Brown / metabolism
  • Adrenergic beta-Agonists / pharmacology
  • Animals
  • Energy Metabolism / drug effects
  • Energy Metabolism / physiology*
  • Humans
  • Thermogenesis / drug effects
  • Thermogenesis / physiology*

Substances

  • Adrenergic beta-Agonists