Effect of different immunosuppressive drugs on immune cells from young and old healthy persons

Gerontology. 2014;60(3):229-38. doi: 10.1159/000356020. Epub 2014 Jan 16.

Abstract

Background: Life expectancy, as well as the average age of patients undergoing solid organ transplantation, increases constantly. Consequently, immunosuppressive therapy is no longer limited to young organ recipients.

Objective: Here, we investigate how different types of immunosuppressive therapy, namely the calcineurin inhibitors cyclosporin A and tacrolimus, as well as the mTOR inhibitor rapamycin, affect the function of immune cells in young and elderly persons.

Methods: Proliferation, cell viability, cytokine production (IL-2, IFN-γ), H2O2 production and telomere length of phytohemagglutinin (PHA)-stimulated human peripheral blood mononuclear cells (PBMCs) of young (n = 13; median age 27 years) and old (n = 19; median age 71 years) healthy donors were analyzed.

Results: The inhibition of proliferation was dampened in PBMCs from elderly donors, especially after incubation with rapamycin. All three immunosuppressive drugs inhibited the production of IL-2 equally well, whereas the production of IFN-γ was less well inhibited by rapamycin. Both calcineurin inhibitors increased H2O2 concentrations after stimulation with PHA and led to a shortening of telomeres in PBMCs from young and old individuals. Rapamycin had only minor effects on H2O2 production and telomere length.

Conclusion: Our results demonstrate that the effects of immunosuppressive drugs on PBMCs differ between young and elderly persons. Calcineurin inhibitors compared to rapamycin have a more pronounced prosenescence effect. These data indicate that specific treatment regimens for the elderly might therefore be considered.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Adult
  • Aged
  • Aged, 80 and over
  • Aging / immunology*
  • Calcineurin Inhibitors / pharmacology
  • Cell Proliferation / drug effects
  • Cyclosporine / pharmacology
  • Female
  • Humans
  • Hydrogen Peroxide / metabolism
  • Immunosuppressive Agents / adverse effects
  • Immunosuppressive Agents / pharmacology*
  • Interferon-gamma / biosynthesis
  • Interleukin-2 / biosynthesis
  • Leukocytes, Mononuclear / cytology
  • Leukocytes, Mononuclear / drug effects*
  • Leukocytes, Mononuclear / immunology*
  • Male
  • Phytohemagglutinins / pharmacology
  • Sirolimus / pharmacology
  • TOR Serine-Threonine Kinases / antagonists & inhibitors
  • Tacrolimus / pharmacology
  • Telomere Shortening / drug effects
  • Young Adult

Substances

  • Calcineurin Inhibitors
  • IL2 protein, human
  • Immunosuppressive Agents
  • Interleukin-2
  • Phytohemagglutinins
  • Interferon-gamma
  • Cyclosporine
  • Hydrogen Peroxide
  • MTOR protein, human
  • TOR Serine-Threonine Kinases
  • Sirolimus
  • Tacrolimus