[Pharmacology of misoprostol (pharmacokinetic data, adverse effects and teratogenic effects)]

J Gynecol Obstet Biol Reprod (Paris). 2014 Feb;43(2):114-22. doi: 10.1016/j.jgyn.2013.11.006. Epub 2014 Jan 17.
[Article in French]

Abstract

Misoprostol is a synthetic analogue of prostaglandin E1. It is used in gynaecology because of its properties of myometrium smooth muscle cells contraction and its effects on the cervix. Misoprostol oral bioavailability is low and several authors have assessed whether the administration by other routes increased its pharmacodynamic effects. This paper summarizes the pharmacokinetic studies after other routes of administration: vaginal, sublingual, buccal or rectal. It also provides an update on its adverse effects and teratogenic effects.

Keywords: Grossesse; Misoprostol; Pharmacocinétique; Pharmacokinectics; Pharmacologie; Pharmacology; Pregnancy; Review; Revue.

Publication types

  • English Abstract

MeSH terms

  • Abnormalities, Drug-Induced / etiology*
  • Abortifacient Agents, Nonsteroidal
  • Abortion, Induced
  • Administration, Buccal
  • Administration, Intravaginal
  • Administration, Rectal
  • Administration, Sublingual
  • Cervical Ripening
  • Cervix Uteri / drug effects
  • Female
  • Humans
  • Misoprostol / administration & dosage
  • Misoprostol / adverse effects*
  • Misoprostol / pharmacokinetics*
  • Oxytocics
  • Pregnancy
  • Uterine Contraction
  • Uterus / drug effects

Substances

  • Abortifacient Agents, Nonsteroidal
  • Oxytocics
  • Misoprostol