Single-entity hydrocodone extended-release capsules in opioid-tolerant subjects with moderate-to-severe chronic low back pain: a randomized double-blind, placebo-controlled study

Pain Med. 2014 Jun;15(6):975-85. doi: 10.1111/pme.12377. Epub 2014 Feb 12.

Abstract

Objective: A single-agent, extended-release formulation of hydrocodone (HC) has been developed for treatment of chronic moderate-to-severe pain. This study was designed to examine the safety and efficacy of HC extended release in opioid-experienced adults with moderate-to-severe chronic low back pain (CLBP).

Methods: This multicenter, enriched enrollment, randomized withdrawal study comprised an open-label conversion/titration phase (≤6 weeks) followed by placebo-controlled, double-blind treatment (12 weeks). During the conversion/titration phase, subjects (N = 510) converted from their current opioid and were titrated to a stabilized dose of HC extended release (20-100 mg every 12 hours). During treatment, subjects (N = 151 per group) received HC extended release or placebo; rescue medication was permitted. The primary efficacy end point was mean change in average pain intensity from baseline to day 85. Response rates (30% pain improvement) and satisfaction (Subject Global Assessment of Medication) were assessed.

Results: Demographic and baseline characteristics were similar between groups. Mean ± SD change in average pain intensity score from baseline to day 85 was significantly lower in the HC extended-release treatment group vs placebo (0.48 ± 1.56 vs 0.96 ± 1.55; P = 0.008). Significantly more responders were in the treatment group (68% vs 31%; P < 0.001). Mean Subject Global Assessment of Medication scores increased significantly (0.8 ± 1.3 vs 0.0 ± 1.4; P < 0.0001), indicating greater satisfaction with HC extended release. The adverse event profile was consistent with other opioids.

Conclusions: Extended-release HC is well tolerated and effective, without acetaminophen-associated risks of liver toxicity, for treatment of CLBP.

Keywords: Chronic Pain; Extended Release; Hydrocodone; Opioids; Randomized Controlled Trial.

Publication types

  • Multicenter Study
  • Randomized Controlled Trial
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Adolescent
  • Adult
  • Aged
  • Analgesics, Opioid / administration & dosage*
  • Chronic Pain / diagnosis
  • Chronic Pain / drug therapy*
  • Delayed-Action Preparations / administration & dosage
  • Double-Blind Method
  • Drug Tolerance*
  • Female
  • Humans
  • Hydrocodone / administration & dosage*
  • Low Back Pain / diagnosis
  • Low Back Pain / drug therapy*
  • Male
  • Middle Aged
  • Pain Measurement / drug effects
  • Pain Measurement / methods
  • Severity of Illness Index*
  • Young Adult

Substances

  • Analgesics, Opioid
  • Delayed-Action Preparations
  • Hydrocodone