Pyrrolidine-mediated direct preparation of (e)-monoarylidene derivatives of homo- and heterocyclic ketones with various aldehydes

Molecules. 2014 Feb 12;19(2):1976-89. doi: 10.3390/molecules19021976.

Abstract

An efficient method for the facile synthesis of (E)-monoarylidene derivatives of homo- and heterocyclic ketones with various aldehydes in the presence of a pyrrolidine organocatalyst has been achieved. A range of α,β-unsaturated ketones were obtained in moderate to high yields (up to 99%). Unlike the Claisen-Schmidt condensation process, the formation of undesired bisarylidene byproducts is not observed. The possible reaction mechanism suggests that the reaction proceeds via a Mannich-elimination sequence.

MeSH terms

  • Aldehydes / chemistry*
  • Catalysis
  • Ketones / chemical synthesis
  • Ketones / chemistry*
  • Molecular Structure
  • Pyrrolidines / chemistry*

Substances

  • Aldehydes
  • Ketones
  • Pyrrolidines
  • pyrrolidine