The chemistry and biological potential of azetidin-2-ones

Eur J Med Chem. 2014 Mar 3:74:619-56. doi: 10.1016/j.ejmech.2014.01.002. Epub 2014 Jan 10.

Abstract

Azetidin-2-ones, commonly referred as β-lactams, represent a unique ring system, with interesting chemistry and great biological potential. Besides its well known antibiotic activity, this ring system exhibits a wide range of activities, attracting the attention of researchers. The biological and pharmacological profile of azetidin-2-ones is reviewed here comprehensively with several examples under fourteen different activity heads. The chemistry and methods of synthesis have also been discussed.

Keywords: Azetidin-2-ones; Pharmacological profile; Synthesis; β-Lactam.

Publication types

  • Review

MeSH terms

  • Anti-Infective Agents / chemical synthesis
  • Anti-Infective Agents / chemistry
  • Anti-Infective Agents / pharmacology
  • Azetidines / chemical synthesis
  • Azetidines / chemistry*
  • Azetidines / pharmacology*
  • Bacteria / drug effects
  • Fungi / drug effects
  • Microbial Sensitivity Tests

Substances

  • 2-azetidinone
  • Anti-Infective Agents
  • Azetidines