2-Acylamido analogues of N-acetylglucosamine prime formation of chitin oligosaccharides by yeast chitin synthase 2

J Biol Chem. 2014 May 2;289(18):12835-41. doi: 10.1074/jbc.M114.550749. Epub 2014 Mar 11.

Abstract

Chitin, a homopolymer of β1,4-linked N-acetylglucosamine (GlcNAc) residues, is a key component of the cell walls of fungi and the exoskeletons of arthropods. Chitin synthases transfer GlcNAc from UDP-GlcNAc to preexisting chitin chains in reactions that are typically stimulated by free GlcNAc. The effect of GlcNAc was probed by using a yeast strain expressing a single chitin synthase, Chs2, by examining formation of chitin oligosaccharides (COs) and insoluble chitin, and by replacing GlcNAc with 2-acylamido analogues of GlcNAc. Synthesis of COs was strongly dependent on inclusion of GlcNAc in chitin synthase incubations, and N,N'-diacetylchitobiose (GlcNAc2) was the major reaction product. Formation of both COs and insoluble chitin was also stimulated by GlcNAc2 and by N-propanoyl-, N-butanoyl-, and N-glycolylglucosamine. MALDI analyses of the COs made in the presence of 2-acylamido analogues of GlcNAc showed they that contained a single GlcNAc analogue and one or more additional GlcNAc residues. These results indicate that Chs2 can use certain 2-acylamido analogues of GlcNAc, and likely free GlcNAc and GlcNAc2 as well, as GlcNAc acceptors in a UDP-GlcNAc-dependent glycosyltransfer reaction. Further, formation of modified disaccharides indicates that CSs can transfer single GlcNAc residues.

Keywords: Carbohydrate Biosynthesis; Chitin; Glycosyltransferases; Polysaccharide; Yeast Physiology.

Publication types

  • Research Support, N.I.H., Extramural

MeSH terms

  • Acetylglucosamine / chemistry
  • Acetylglucosamine / metabolism*
  • Acetylglucosamine / pharmacology
  • Cell Membrane / chemistry
  • Cell Membrane / drug effects
  • Cell Membrane / metabolism
  • Chitin / biosynthesis*
  • Chitin / chemistry
  • Chitin Synthase / genetics
  • Chitin Synthase / metabolism*
  • Disaccharides / chemistry
  • Disaccharides / metabolism
  • Dose-Response Relationship, Drug
  • Glucose / pharmacology
  • Mutation
  • Oligosaccharides / biosynthesis*
  • Oligosaccharides / chemistry
  • Saccharomyces cerevisiae / chemistry
  • Saccharomyces cerevisiae / genetics
  • Saccharomyces cerevisiae / metabolism
  • Saccharomyces cerevisiae Proteins / genetics
  • Saccharomyces cerevisiae Proteins / metabolism*
  • Spectrometry, Mass, Matrix-Assisted Laser Desorption-Ionization

Substances

  • Disaccharides
  • Oligosaccharides
  • Saccharomyces cerevisiae Proteins
  • Chitin
  • N,N-diacetylchitobiose
  • Chitin Synthase
  • Chs2 protein, S cerevisiae
  • Glucose
  • Acetylglucosamine