Conversion of pyridine N-oxides to tetrazolopyridines

J Org Chem. 2014 Apr 4;79(7):3249-54. doi: 10.1021/jo500231m. Epub 2014 Mar 21.

Abstract

An efficient and convenient procedure for the conversion of pyridine N-oxides to tetrazolopyridines by treatment with 4-toluene sulfonyl chloride and sodium azide in toluene at elevated temperature is described.