Lucimycin, an antifungal peptide from the therapeutic maggot of the common green bottle fly Lucilia sericata

Biol Chem. 2014 Jun;395(6):649-56. doi: 10.1515/hsz-2013-0263.

Abstract

We report the identification, cloning, heterologous expression and functional characterization of a novel antifungal peptide named lucimycin from the common green bottle fly Lucilia sericata. The lucimycin cDNA was isolated from a library of genes induced during the innate immune response in L. sericata larvae, which are used as therapeutic maggots. The peptide comprises 77 amino acid residues with a molecular mass of 8.2 kDa and a pI of 6.6. It is predicted to contain a zinc-binding motif and to form a random coil, lacking β-sheets or other secondary structures. Lucimycin was active against fungi from the phyla Ascomycota, Basidiomycota and Zygomycota, in addition to the oomycete Phytophtora parasitica, but it was inactive against bacteria. A mutant version of lucimycin, lacking the four C-terminal amino acid residues, displayed 40-fold lower activity. The activity of lucimycin against a number of highly-destructive plant pathogens could be exploited to produce transgenic crops that are resistant against fungal diseases.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Antifungal Agents / metabolism*
  • Larva
  • Lucensomycin / metabolism*
  • Peptides / metabolism*
  • Sequence Analysis, Protein

Substances

  • Antifungal Agents
  • Peptides
  • Lucensomycin