Molecular dosimetry of endogenous and exogenous O(6)-methyl-dG and N7-methyl-G adducts following low dose [D3]-methylnitrosourea exposures in cultured human cells

Chem Res Toxicol. 2014 Apr 21;27(4):480-2. doi: 10.1021/tx5000602. Epub 2014 Mar 26.

Abstract

For DNA-reactive chemicals, a low dose linear assessment of cancer risk is the science policy default. In the present study, we quantitated the endogenous and exogenous N7-methyl-G and O(6)-methyl-dG adducts in human lymphoblastoid cells exposed to low dose [D3]-methylnitrosourea. Endogenous amounts of both adducts remained nearly constant, while the exogenous adducts showed linear dose-responses. The data show that O(6)-methyl-dG adducts ≥1.8/10(8) dG correlated with published studies that demonstrated significant increases of mutations under these conditions. The combined results do not support linear extrapolations to zero when data are available for science-based regulations.

Publication types

  • Research Support, N.I.H., Extramural

MeSH terms

  • Cells, Cultured
  • Deoxyguanosine / analogs & derivatives*
  • Deoxyguanosine / metabolism
  • Dose-Response Relationship, Drug
  • Guanine / analogs & derivatives*
  • Guanine / metabolism
  • Humans
  • Methylnitrosourea / administration & dosage
  • Methylnitrosourea / pharmacology*

Substances

  • Guanine
  • 7-methylguanine
  • Methylnitrosourea
  • O(6)-methyl-2'-deoxyguanosine
  • Deoxyguanosine