Sulphonylurea usage in melioidosis is associated with severe disease and suppressed immune response

PLoS Negl Trop Dis. 2014 Apr 24;8(4):e2795. doi: 10.1371/journal.pntd.0002795. eCollection 2014 Apr.

Abstract

Background: Melioidosis is a problem in the developing tropical regions of Southeast Asia and Northern Australia where the the Gram negative saprophytic bacillus Burkholderia pseudomallei is endemic with the risk of fulminant septicaemia. While diabetes mellitus is a well-established risk factor for melioidiosis, little is known if specific hypoglycemic agents may differentially influence the susceptibility and clinical course of infection with B. pseudomallei (Bp).

Methodology/principal findings: In this cohort study, patients with pre-existing diabetes and melioidosis were retrospectively studied.

Outcome measures: mortality, length of stay and development of complications (namely hypotension, intubation, renal failure and septicaemia) were studied in relation to prior diabetic treatment regimen. Peripheral blood mononuclear cells (PBMC) from diabetic patients and healthy PBMC primed with metformin, glyburide and insulin were stimulated with purified Bp antigens in vitro. Immune response and specific immune pathway mediators were studied to relate to the clinical findings mechanistically. Of 74 subjects, 44 (57.9%) had sulphonylurea-containing diabetic regimens. Patient receiving sulphonylureas had more severe septic complications (47.7% versus 16.7% p = 0.006), in particular, hypotension requiring intropes (p = 0.005). There was also a trend towards increased mortality in sulphonylurea-users (15.9% versus 3.3% p = 0.08). In-vitro, glyburide suppressed inflammatory cytokine production in a dose-dependent manner. An effect of the drug was the induction of IL-1R-associated kinase-M at the level of mRNA transcription.

Conclusion/significance: Sulphonylurea treatment results in suppression of host inflammatory response and may put patients at higher risk for adverse outcomes in melioidosis.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Asia, Southeastern
  • Australia
  • Cohort Studies
  • Diabetes Complications / epidemiology
  • Diabetes Mellitus / drug therapy
  • Female
  • Humans
  • Hypoglycemic Agents / adverse effects*
  • Hypoglycemic Agents / therapeutic use*
  • Length of Stay
  • Male
  • Melioidosis / complications
  • Melioidosis / immunology*
  • Melioidosis / mortality
  • Melioidosis / pathology*
  • Middle Aged
  • Retrospective Studies
  • Sepsis / mortality
  • Sepsis / pathology
  • Sulfonylurea Compounds / adverse effects*
  • Sulfonylurea Compounds / therapeutic use*
  • Survival Analysis
  • Treatment Outcome

Substances

  • Hypoglycemic Agents
  • Sulfonylurea Compounds

Grants and funding

This study was funded by the MINDEF-NUS Joint Applied R&D Cooperation (JPP) Programme as well as the following grants awarded to Louis Chai: New Investigator Grant (NIG), Clinician Scientist Award (CSA), Individual Research Grant (IRG) and Bedside & Bench (B&B) grants of the National Medical Research Council (NMRC), Singapore, and the National Kidney Foundation, Singapore. The funders had no role in study design, data collection and analysis, decision to publish, or preparation of the manuscript.