Huaier suppresses proliferation and induces apoptosis in human pulmonary cancer cells via upregulation of miR-26b-5p

FEBS Lett. 2014 Jun 5;588(12):2107-14. doi: 10.1016/j.febslet.2014.04.044. Epub 2014 May 8.

Abstract

Various studies have reported that Huaier possesses anti-tumor effects. However, the mechanisms are not completely elucidated. Here, we found 66 differentially expressed miRNAs in Huaier-treated pulmonary adenocarcinoma A549 cells, with upregulation of miR-26b-5p. Transfection of A549 cells with miR-26b-5p mimic inhibited proliferation and induced apoptosis, while transfection of Huaier-treated A549 cells with a miR-26b-5p inhibitor reversed the effects of Huaier. EZH2 was verified as the target of miR-26b-5p. Thus, our findings indicate that Huaier might suppress proliferation and induce apoptosis in lung cancer cells via a miR-26b-5p-EZH2-mediated approach, which provides a new perspective for understanding the anti-tumor effects of Huaier.

Keywords: Apoptosis; EZH2; Huaier; Lung cancer; Proliferation; miR-26b-5p.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Antineoplastic Agents / pharmacology*
  • Apoptosis / drug effects*
  • Base Sequence
  • Cell Line, Tumor
  • Cell Proliferation / drug effects
  • Enhancer of Zeste Homolog 2 Protein
  • Humans
  • Lung Neoplasms / pathology*
  • MicroRNAs / genetics*
  • Polycomb Repressive Complex 2 / genetics
  • Proto-Oncogene Proteins c-bcl-2 / genetics
  • Trametes / chemistry*
  • Trametes / physiology
  • Up-Regulation / drug effects*
  • beta Catenin / genetics

Substances

  • Antineoplastic Agents
  • MIRN26A microRNA, human
  • MicroRNAs
  • Proto-Oncogene Proteins c-bcl-2
  • beta Catenin
  • EZH2 protein, human
  • Enhancer of Zeste Homolog 2 Protein
  • Polycomb Repressive Complex 2