Sucrose/Glucose molecular alloys by cryomilling

J Pharm Sci. 2014 Jul;103(7):2098-2106. doi: 10.1002/jps.24027. Epub 2014 May 27.

Abstract

We report here for the first time a series of amorphous sucrose/glucose molecular alloys prepared by cryomilling. Differential scanning calorimetry, X-ray powder diffraction and solution proton nuclear magnetic resonance showed that cryomilling drives a direct transformation from a two-phase mixture of crystalline sucrose and glucose, to a single-phase amorphous sucrose/glucose molecular alloy. The molecular alloys displayed a single Tg which varied linearly with composition. The effect of atmospheric moisture and the possibility of localised melting of the material because of milling-related friction were also discussed.

Keywords: X-ray powder diffractometry; amorphous; calorimetry (DSC); materials science; milling.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Calorimetry, Differential Scanning
  • Crystallization
  • Excipients / chemistry*
  • Glucose / chemistry*
  • Phase Transition*
  • Sucrose / chemistry*
  • Transition Temperature
  • X-Ray Diffraction

Substances

  • Excipients
  • Sucrose
  • Glucose