Thalidomide ameliorates inflammation and vascular injury but aggravates tubular damage in the irradiated mouse kidney

Int J Radiat Oncol Biol Phys. 2014 Jul 1;89(3):599-606. doi: 10.1016/j.ijrobp.2014.03.039.

Abstract

Purpose: The late side effects of kidney irradiation include vascular damage and fibrosis, which are promoted by an irradiation-induced inflammatory response. We therefore treated kidney-irradiated mice with the anti-inflammatory and angiogenesis-modulating drug thalidomide in an attempt to prevent the development of late normal tissue damage and radiation nephropathy in the mouse kidney.

Methods and materials: Kidneys of C57Bl/6 mice were irradiated with a single dose of 14 Gy. Starting from week 16 after irradiation, the mice were fed with thalidomide-containing chow (100 mg/kg body weight/day). Gene expression and kidney histology were analyzed at 40 weeks and blood samples at 10, 20, 30, and 40 weeks after irradiation.

Results: Thalidomide improved the vascular structure and vessel perfusion after irradiation, associated with a normalization of pericyte coverage. The drug also reduced infiltration of inflammatory cells but could not suppress the development of fibrosis. Irradiation-induced changes in hematocrit and blood urea nitrogen levels were not rescued by thalidomide. Moreover, thalidomide worsened tubular damage after irradiation and also negatively affected basal tubular function.

Conclusions: Thalidomide improved the inflammatory and vascular side effects of kidney irradiation but could not reverse tubular toxicity, which probably prevented preservation of kidney function.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Angiogenesis Modulating Agents / adverse effects
  • Angiogenesis Modulating Agents / pharmacology*
  • Animals
  • Anti-Inflammatory Agents / adverse effects
  • Anti-Inflammatory Agents / pharmacology*
  • Female
  • Fibrosis
  • Genes, sis / drug effects
  • Glomerular Filtration Rate / drug effects
  • Glomerular Filtration Rate / radiation effects
  • Kidney / blood supply
  • Kidney / drug effects
  • Kidney / pathology
  • Kidney / radiation effects*
  • Kidney Tubules / drug effects*
  • Kidney Tubules / radiation effects
  • Mice
  • Mice, Inbred C57BL
  • Nephritis / pathology
  • Nephritis / prevention & control
  • Radiation Injuries, Experimental / prevention & control*
  • Thalidomide / adverse effects
  • Thalidomide / pharmacology*

Substances

  • Angiogenesis Modulating Agents
  • Anti-Inflammatory Agents
  • Thalidomide