Influence of repetitive contrast agent injections on functional and molecular ultrasound measurements

Ultrasound Med Biol. 2014 Oct;40(10):2468-75. doi: 10.1016/j.ultrasmedbio.2014.04.010. Epub 2014 Jul 9.

Abstract

Quantitative contrast-enhanced ultrasound plays an important role in tumor characterization and treatment assessment. Besides established functional ultrasound techniques, ultrasound molecular imaging using microbubbles targeted to disease-associated markers is increasingly being applied in pre-clinical studies. Often, repeated injections of non-targeted or targeted microbubbles during the same imaging session are administered. However, the influence of repeated injections on the accuracy of the quantitative data is unclear. Therefore, in tumor-bearing mice, we investigated the influence of multiple injections of non-targeted microbubbles (SonoVue) on time to peak and peak enhancement in liver and tumor tissue and of vascular endothelial growth factor receptor 2 (VEGFR2)-targeted contrast agents (MicroMarker) on specific tumor accumulation. We found significantly decreasing values for time to peak and a tendency for increased values for peak enhancement after multiple injections. Repeated injections of VEGFR2-targeted microbubbles led to significantly increased tumor accumulation, which may result from the exposure of additional binding sites at endothelial surfaces caused by mechanical forces from destroyed microbubbles.

Keywords: Cancer; Contrast-enhanced ultrasound; Molecular ultrasound; Multiple injections; Peak enhancement; Quantitative imaging; Reproducibility; SonoVue; Time to peak; VEGFR2; Vascular endothelial growth factor receptor 2.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Carcinoma, Squamous Cell / diagnostic imaging*
  • Contrast Media / administration & dosage*
  • Contrast Media / pharmacokinetics
  • Female
  • Image Enhancement / methods
  • Injections
  • Liver / metabolism*
  • Mice
  • Mice, Nude
  • Microbubbles
  • Molecular Imaging / methods*
  • Phospholipids / administration & dosage*
  • Phospholipids / pharmacokinetics
  • Reproducibility of Results
  • Sensitivity and Specificity
  • Sulfur Hexafluoride / administration & dosage*
  • Sulfur Hexafluoride / pharmacokinetics
  • Ultrasonography
  • Vascular Endothelial Growth Factor Receptor-2 / metabolism

Substances

  • Contrast Media
  • Phospholipids
  • contrast agent BR1
  • Vascular Endothelial Growth Factor Receptor-2
  • Sulfur Hexafluoride