Access to novel functionalized trifluoromethyl β-lactams by ring expansion of aziridines

Org Biomol Chem. 2014 Sep 7;12(33):6345-8. doi: 10.1039/c4ob01262c.

Abstract

From carboxylic acid trifluoromethyl aziridines, halogeno β-lactams were obtained stereoselectively by ring expansion. Different conditions such as radical, organometallic reactions allowed easy and selective access to CF3-β-lactams substituted at the C-3 position.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Aziridines / chemistry*
  • Lactams / chemical synthesis*
  • Lactams / chemistry
  • Molecular Structure

Substances

  • Aziridines
  • Lactams