Retreatment of men with metastatic castrate-resistant prostate cancer with abiraterone

Prostate. 2014 Oct;74(14):1462-4. doi: 10.1002/pros.22861. Epub 2014 Aug 11.

Abstract

Background: Abiraterone acetate (AA), oral CYP17 inhibitor, is an active agent in the treatment of metastatic castrate-resistant prostate cancer (mCRPC).

Methods: We (R.L.A and N.A) retrospectively evaluated outcome in 12 men who were re-treated with AA following prior treatment with AA at the Princess Margaret Cancer Centre.

Results: All men were heavily pre-treated for mCRPC with a median of four prior lines of therapy, one of which was AA (given either pre- or post-chemotherapy). Eleven out of 12 (92%) men stopped their first treatment course of AA due to progression and one stopped for financial reasons. Seven men had a PSA decrease ≥50% following their first AA treatment, of which three (46%) had a PSA decrease ≥50% to AA re-treatment. The responses to AA re-treatment were generally short-lived with a median biochemical progression-free survival of 2.3 months and median treatment duration of 3.2 months. No PSA responses to AA re-treatment were seen in five men who did not have an initial PSA response to AA.

Conclusions: Our data suggest that AA re-challenge may have limited benefit in select men with mCRPC, and warrants further formal research.

Keywords: abiraterone; mCRPC; re-challenge.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Abiraterone Acetate
  • Aged
  • Aged, 80 and over
  • Androstadienes / therapeutic use*
  • Enzyme Inhibitors / therapeutic use*
  • Humans
  • Male
  • Middle Aged
  • Prostatic Neoplasms, Castration-Resistant / drug therapy*
  • Prostatic Neoplasms, Castration-Resistant / enzymology
  • Retrospective Studies
  • Steroid 17-alpha-Hydroxylase / antagonists & inhibitors
  • Steroid 17-alpha-Hydroxylase / metabolism

Substances

  • Androstadienes
  • Enzyme Inhibitors
  • Steroid 17-alpha-Hydroxylase
  • Abiraterone Acetate