TLR4-dependent activation of dendritic cells by an HMGB1-derived peptide adjuvant

J Transl Med. 2014 Aug 14:12:211. doi: 10.1186/1479-5876-12-211.

Abstract

High mobility group box protein 1 (HMGB1) acts as an endogenous danger molecule that is released from necrotic cells and activated macrophages. We have previously shown that peptide Hp91, whose sequence corresponds to an area within the B-Box domain of HMGB1, activates dendritic cells (DCs) and acts as an adjuvant in vivo. Here we investigated the underlying mechanisms of Hp91-mediated DC activation. Hp91-induced secretion of IL-6 was dependent on clathrin- and dynamin-driven endocytosis of Hp91 and mediated through a MyD88- and TLR4-dependent pathway involving p38 MAPK and NFκB. Endosomal TLR4 has been shown to activate the MyD88-independent interferon pathway. Hp91-induced activation of pIRF3 and IL-6 secretion was reduced in IFNαβR knockout DCs, suggesting an amplification loop via the IFNαβR. These findings elucidate the mechanisms by which Hp91 acts as immunostimulatory peptide and may serve as a guide for the future development of synthetic Th1-type peptide adjuvants for vaccines.

Publication types

  • Research Support, N.I.H., Extramural
  • Research Support, Non-U.S. Gov't
  • Research Support, U.S. Gov't, Non-P.H.S.

MeSH terms

  • Adjuvants, Immunologic / pharmacology*
  • Animals
  • Cells, Cultured
  • Dendritic Cells / drug effects*
  • Dendritic Cells / immunology*
  • Dendritic Cells / metabolism
  • Female
  • HMGB1 Protein / chemistry
  • HMGB1 Protein / immunology
  • HMGB1 Protein / pharmacology*
  • Humans
  • Immunotherapy, Adoptive / methods
  • Mice
  • Mice, Inbred C57BL
  • Mice, Knockout
  • Peptide Fragments / immunology
  • Peptide Fragments / pharmacology*
  • Protein Structure, Tertiary
  • Signal Transduction / drug effects
  • Signal Transduction / genetics
  • Signal Transduction / immunology
  • Toll-Like Receptor 4 / genetics
  • Toll-Like Receptor 4 / physiology*

Substances

  • Adjuvants, Immunologic
  • HMGB1 Protein
  • Peptide Fragments
  • Tlr4 protein, mouse
  • Toll-Like Receptor 4